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Biochemical Rat MASP2 Assay from US Patent US20240010684: "MASP INHIBITORY COMPOUNDS AND USES THEREOF"
Assay data:20 Active, 20 Activity ≤ 1 µM, 20 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Depositor
Biochemical Rat MASP1 Assay from US Patent US20240010684: "MASP INHIBITORY COMPOUNDS AND USES THEREOF"
Assay data:21 Active, 21 Activity ≤ 1 µM, 21 Tested
Biological and Stability Data from US Patent US11458151: "Toll-like receptor ligands"
Assay data:8 Active, 5 Activity ≤ 1 nM, 8 Activity ≤ 1 µM, 8 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Radioligand Binding Assay on Rat TAAR1 from US Patent US11697636: "Substituted benzamides"
Assay data:313 Active, 31 Activity ≤ 1 nM, 305 Activity ≤ 1 µM, 314 Tested
Competitive Radioligand Binding Assay from US Patent US11691947: "Isoindoline compositions and methods for treating neurodegenerative disease"
Assay data:81 Active, 3 Activity ≤ 1 nM, 79 Activity ≤ 1 µM, 93 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Binding to Nicotinic Receptor Subtypes from US Patent US11667638: "4-substitued cytisine analogues"
Assay data:50 Active, 3 Activity ≤ 1 nM, 50 Activity ≤ 1 µM, 50 Tested
Steroid Inhibition of TBPS Binding from US Patent US11542297: "Compositions and methods for treating CNS disorders"
Assay data:214 Active, 230 Activity ≤ 1 µM, 230 Tested
Radioligand Competition Binding Assay from US Patent US11518754: "Radiolabeled pharmaceuticals and methods of making and using same"
Assay data:10 Active, 2 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
Steroid Inhibition of TBPS Binding from US Patent US11147877: "Compositions and methods for treating CNS disorders"
Assay data:11 Active, 17 Activity ≤ 1 µM, 17 Tested
Rat FAAH Inhibition Assay from US Patent US10918640: "Azetidine derivatives"
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Enzyme Inhibition Assay from US Patent US10759791: "Mammalian and bacterial nitric oxide synthase inhibitors"
Assay data:24 Active, 21 Activity ≤ 1 µM, 24 Tested
Screen Quest Fluo-8 No Wash Calcium Assay Kit from US Patent US10669267: "Substituted N-[2-(4-phenoxypiperidin-1-yl)-2-(1,3-thiazol-5-yl)ethyl]benzamide and N-[2-(4-benzyloxypiperidin-1-yl)-2-(1,3-thiazol-5-yl)ethyl]benzamide derivatives P2X7 receptor antagonists"
Assay data:39 Active, 32 Activity ≤ 1 µM, 39 Tested
Fluorescent Assay from US Patent US10662159: "ABHD6 and dual ABHD6/MGL inhibitors and their uses"
Assay data:30 Activity ≤ 1 µM, 30 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
FLIPR Tetra Assay from US Patent US10597383: "Bicyclic proline compounds"
Assay data:35 Active, 35 Activity ≤ 1 µM, 35 Tested
Ca2+ Flux Assay from US Patent US10538491: "4,5-substituted picolinamide and picolinonitrile metabotropic glutamate receptor 2 negative allosteric modulators"
Assay data:95 Active, 41 Activity ≤ 1 µM, 153 Tested
Receptor Binding Assay from US Patent US10501452: "Lactam compound derivative and application thereof"
Assay data:23 Active, 23 Activity ≤ 1 µM, 23 Tested
In Vitro Rat FAAH Radiometric Assay from US Patent US10435355: "Inhibitors of fatty acid amide hydrolase (FAAH) enzyme with improved oral bioavailability and their use as medicaments"
Assay data:13 Active, 3 Activity ≤ 1 nM, 13 Activity ≤ 1 µM, 13 Tested
Rat FAAH Inhibition Assay from US Patent US10383871: "Azetidine derivatives"
Biological Assay from US Patent US10364234: "Pyridinecarboxamide derivatives, preparation method thereof and pharmaceutical uses thereof"
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
FLIPR Assay from US Patent US9464084: "P2X7 modulators"
Assay data:277 Active, 2 Activity ≤ 1 nM, 237 Activity ≤ 1 µM, 293 Tested
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