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Inhibition of LOX and LOXL1-4 from US Patent US20230349907: "BIOPROBES FOR LYSYL OXIDASES AND USES THEREOF"
Assay data:10 Active, 16 Activity ≤ 1 µM, 16 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
LOX Enzyme Activity Assay from US Patent US11608330: "Methylamine derivatives as lysysl oxidase inhibitors for the treatment of cancer"
Assay data:86 Active, 28 Activity ≤ 1 µM, 89 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Protein Kinase Assay Condition B (Thiol-Free Conditions) from US Patent US11447493: "Inhibitors of cyclin-dependent kinases"
Assay data:14 Active, 14 Activity ≤ 1 µM, 14 Tested
Protein Kinase Assay Condition A (Thiol Containing Conditions) from US Patent US11447493: "Inhibitors of cyclin-dependent kinases"
Assay data:79 Active, 64 Activity ≤ 1 µM, 95 Tested
Chromogenic Enzyme Activity Assays from US Patent US11149067: "Tailored cyclodepsipeptides as potent non-covalent serine protease inhibitors"
Assay data:31 Active, 19 Activity ≤ 1 µM, 33 Tested
Enzyme Inhibition Assay from US Patent US10759791: "Mammalian and bacterial nitric oxide synthase inhibitors"
Assay data:24 Active, 21 Activity ≤ 1 µM, 24 Tested
Xanthine Oxidase (XO) Assay from Article 10.1111/cbdd.12686: "Development of 2-(Substituted Benzylamino)-4-Methyl-1, 3-Thiazole-5-Carboxylic Acid Derivatives as Xanthine Oxidase Inhibitors and Free Radical Scavengers."
Assay data:4 Active, 1 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Cyclooxygenase Assay from Article 10.1111/cbdd.12457: "Synthesis, Molecular Modeling, and Biological Evaluation of Novel 1, 3-Diphenyl-2-propen-1-one Based Pyrazolines as Anti-inflammatory Agents."
Assay data:16 Active, 4 Activity ≤ 1 µM, 19 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
In vitro Cyclooxygenase Inhibition Assay from Article 10.1111/cbdd.12435: "1,2-Diaryl-2-hydroxyiminoethanones as dual COX-1 and -amyloid aggregation inhibitors: biological evaluation and in silico study."
Assay data:4 Active, 2 Activity ≤ 1 µM, 7 Tested
In Vitro Isomerase Inhibition Assay from US Patent US10188615: "Alkoxy compounds for disease treatment"
Assay data:167 Active, 140 Activity ≤ 1 µM, 169 Tested
Inhibition Assay from US Patent US11098045: "Haloallylamine indole and azaindole derivative inhibitors of lysyl oxidases and uses thereof"
Assay data:116 Active, 116 Activity ≤ 1 µM, 116 Tested
Fluorescence Polarization Assay from US Patent US11028041: "Second generation GRP94-selective inhibitors"
Assay data:16 Active, 12 Activity ≤ 1 µM, 18 Tested
LOX Enzyme Activity Assay from US Patent US10807974: "Methylamine derivatives as lysysl oxidase inhibitors for the treatment of cancer"
Assay data:85 Active, 28 Activity ≤ 1 µM, 88 Tested
Binding Inhibition Assay from US Patent US10759796: "CXCR4 inhibitors and uses thereof"
Assay data:126 Active, 138 Activity ≤ 1 µM, 138 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Inhibition Assay from US Patent US10717734: "Indole and azaindole haloallylamine derivative inhibitors of lysyl oxidases and uses thereof"
Assay data:44 Tested
SummaryRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition Assay from US Patent US10717733: "Haloallylamine indole and azaindole derivative inhibitors of lysyl oxidases and uses thereof"
In Vitro Isomerase Inhibition Assay from US Patent US10639286: "Alkoxy compounds for disease treatment"
Assay data:166 Active, 139 Activity ≤ 1 µM, 172 Tested
Fluorescence Polarization Assay from US Patent US10464907: "Compound having HSP90 inhibitory activity or pharmaceutically acceptable salt thereof, and medical use thereof"
Assay data:29 Active, 23 Activity ≤ 1 µM, 29 Tested
Inhibition Assay from US Patent US10383835: "Treatment of inflammatory disorders in non-human mammals"
Assay data:25 Active, 6 Activity ≤ 1 nM, 20 Activity ≤ 1 µM, 25 Tested
In Vitro Measurements of porcine D-Amino Acid Oxidase (DAAO) Activities from US Patent US10336724: "D-amino acid oxidase inhibitors and therapeutic uses thereof"
Assay data:14 Active, 11 Activity ≤ 1 µM, 19 Tested
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