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BIOLOGICAL ASSAYS from US Patent US10221163: "Metallo-beta-lactamase inhibitors"
Assay data:491 Active, 461 Activity ≤ 1 nM, 491 Activity ≤ 1 µM, 491 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Antibacterial activity against Klebsiella pneumoniae ATCC BAA-2146 assessed as inhibition in bacterial growth incubated for 20 to 24 hrs by CLSI based broth microdilution method
Assay data:21 Tested
SummaryPubMed Citation
Antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as inhibition in bacterial growth incubated for 20 to 24 hrs by CLSI based broth microdilution method
Antibacterial activity against Klebsiella pneumoniae ATCC 10031 assessed as inhibition in bacterial growth incubated for 20 to 24 hrs by CLSI based broth microdilution method
Antibacterial activity against Klebsiella pneumoniae ATCC BAA-1705 assessed as inhibition in bacterial growth incubated for 20 to 24 hrs by CLSI based broth microdilution method
Assay data:19 Tested
Antimicrobial activity against Klebsiella pneumoniae 02-63 assessed as reduction in microbial cell growth incubated for 16 to 18 hrs by Mueller-Hinton broth based microdilution method
Assay data:1 Tested
Antibacterial activity against Klebsiella pneumoniae BAA 1705 assessed as bacterial growth inhibition incubated for 16 to 18 hrs by CLSI based antibiotic susceptibility testing method
Assay data:43 Tested
Antibacterial activity against Klebsiella pneumoniae assessed as reduction in bacterial growth by CLSI protocol based method
Assay data:22 Tested
Antibacterial activity against pandrug-resistant Klebsiella pneumoniae MS6671 assessed as reduction in bacterial growth by microbroth dilution assay
Assay data:14 Tested
Antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as reduction in bacterial growth by microbroth dilution assay
Antibacterial activity against Klebsiella pneumoniae ATCC 33495 assessed as reduction in bacterial growth by microbroth dilution assay
Potentiation of novobiocin induced antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as decrease in bacterial growth at 0.4 uM incubated for 18 hrs in presence of novobiocin by two fold serial dilution assay
Assay data:15 Active, 15 Tested
SummaryCompounds, ActivePubMed Citation
Potentiation of fusidic acid induced antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as decrease in bacterial growth at 0.4 uM incubated for 18 hrs in presence of fusidic acid by two fold serial dilution assay
Potentiation of erythromycin induced antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as decrease in bacterial growth at 0.4 uM incubated for 18 hrs in presence of erythromycin by two fold serial dilution assay
Antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as inhibition of bacterial growth incubated for 18 hrs in presence of rifampicin with calcium and Mg2+ broth media by two fold serial dilution assay
Antibacterial activity against Klebsiella pneumoniae ATCC 700603 assessed as inhibition of bacterial growth incubated for 18 hrs by two fold serial dilution assay
Assay data:3 Active, 33 Tested
Inhibition of Metallo-beta-lactamase NDM-1 (unknown origin) using nitrocefin as substrate incubated for 5 to 10 mins by spectramax reader analysis
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Antimicrobial activity against Klebsiella pneumoniae assessed as reduction in bacterial growth incubated for 20 hrs by broth microdilution analysis
Assay data:15 Tested
Antibacterial activity against multidrug-resistant Klebsiella pneumoniae clinical isolates assessed as inhibition of bacterial growth at 20 uM by broth microdilution method
Assay data:3 Tested
Antibacterial activity against Klebsiella pneumoniae assessed as inhibition of bacterial growth
Assay data:24 Tested
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