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Functional Calcium Imaging Assay from Article 10.1074/jbc.M114.573162: "ORA1, a zebrafish olfactory receptor ancestral to all mammalian V1R genes, recognizes 4-hydroxyphenylacetic acid, a putative reproductive pheromone."
Assay data:1 Active, 11 Tested
SummaryCompounds, ActivePubMed Citation
Drug uptake in zebrafish embryo assessed as penetration depth at 20 uM treated for 20 mins by two-photon based fluorescence microscopy
Assay data:1 Tested
SummaryPubMed Citation
Prodrug activation in zebrafish assessed as NO release by measuring red fluorescence signal at 20 uM incubated for 20 mins by dRB-OPD staining based fluorescence microscopy
Prodrug activation in zebrafish assessed as green fluorescence signal at 20 uM incubated for 20 mins by fluorescence microscopy
Induction of apoptosis in zebrafish embryo assessed as increase intracellular ROS level at 0.01 to 1 uM measured by DCFH-DA dye based flow cytometric analysis
Assay data:1 Active, 1 Tested
Competitive inhibition of N-terminal His-SUMO tagged zebra fish recombinant HDAC6 catalytic domain 2 transfected with pET28b(+) vector in Escherichia coli BL21 (DE3) RILP cells incubated for 10 mins followed by addition of FITC-M344 measured af ter 10 mins by fluorescence polarization assay
Assay data:9 Active, 8 Activity ≤ 1 µM, 9 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in brain at 0.7 uM measured after 14 days by microscopy
Assay data:1 Active, 2 Tested
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in brain at 8.9 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in muscle at 0.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in heart at 0.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in yolk sac at 0.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in brain at 0.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in muscle at 1.5 uM measured after 14 days by microscopy
Assay data:2 Active, 3 Tested
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in heart at 1.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in yolk sac at 1.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in brain at 1.5 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARgamma in transgenic zebrafish assessed as increase in GFP expression in muscle at 1 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARgamma in transgenic zebrafish assessed as increase in GFP expression in CNS at 1 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARgamma in transgenic zebrafish assessed as increase in GFP expression in tail bud at 0.1 uM measured after 14 days by microscopy
In vivo agonist activity at human GFP-tagged PPARalpha in transgenic zebrafish assessed as increase in GFP expression in muscle at 5 uM measured after 14 days by microscopy
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