Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Inhibition of LOX and LOXL1-4 from US Patent US20230349907: "BIOPROBES FOR LYSYL OXIDASES AND USES THEREOF"
Assay data:10 Active, 16 Activity ≤ 1 µM, 16 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Protein Kinase Assay Condition B (Thiol-Free Conditions) from US Patent US11447493: "Inhibitors of cyclin-dependent kinases"
Assay data:14 Active, 14 Activity ≤ 1 µM, 14 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Protein Kinase Assay Condition A (Thiol Containing Conditions) from US Patent US11447493: "Inhibitors of cyclin-dependent kinases"
Assay data:79 Active, 64 Activity ≤ 1 µM, 95 Tested
Chromogenic Enzyme Activity Assays from US Patent US11149067: "Tailored cyclodepsipeptides as potent non-covalent serine protease inhibitors"
Assay data:31 Active, 19 Activity ≤ 1 µM, 33 Tested
Enzyme Inhibition Assay from US Patent US10759791: "Mammalian and bacterial nitric oxide synthase inhibitors"
Assay data:24 Active, 21 Activity ≤ 1 µM, 24 Tested
Xanthine Oxidase (XO) Assay from Article 10.1111/cbdd.12686: "Development of 2-(Substituted Benzylamino)-4-Methyl-1, 3-Thiazole-5-Carboxylic Acid Derivatives as Xanthine Oxidase Inhibitors and Free Radical Scavengers."
Assay data:4 Active, 1 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
In Vitro Isomerase Inhibition Assay from US Patent US10188615: "Alkoxy compounds for disease treatment"
Assay data:167 Active, 140 Activity ≤ 1 µM, 169 Tested
Inhibition Assay from US Patent US11098045: "Haloallylamine indole and azaindole derivative inhibitors of lysyl oxidases and uses thereof"
Assay data:116 Active, 116 Activity ≤ 1 µM, 116 Tested
Binding Inhibition Assay from US Patent US10759796: "CXCR4 inhibitors and uses thereof"
Assay data:126 Active, 138 Activity ≤ 1 µM, 138 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µM
Inhibition Assay from US Patent US10717734: "Indole and azaindole haloallylamine derivative inhibitors of lysyl oxidases and uses thereof"
Assay data:44 Tested
SummaryRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition Assay from US Patent US10717733: "Haloallylamine indole and azaindole derivative inhibitors of lysyl oxidases and uses thereof"
In Vitro Isomerase Inhibition Assay from US Patent US10639286: "Alkoxy compounds for disease treatment"
Assay data:166 Active, 139 Activity ≤ 1 µM, 172 Tested
Fluorescence Polarization Assay from US Patent US10464907: "Compound having HSP90 inhibitory activity or pharmaceutically acceptable salt thereof, and medical use thereof"
Assay data:29 Active, 23 Activity ≤ 1 µM, 29 Tested
Inhibtion Assay from US Patent US9493447: "Optically active PDE10 inhibitor"
Assay data:3 Active, 2 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 3 Tested
SOD Assay (Kinetic Analysis) from Article 10.3109/14756366.2012.680063: "Interaction of superoxide dismutase with the glycine zipper regions of -amyloid peptides: is there an implication towards Alzheimer's disease and oxidative stress?"
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Depositor
SOD Assay (Fluorimetric Analysis) from Article 10.3109/14756366.2012.680063: "Interaction of superoxide dismutase with the glycine zipper regions of -amyloid peptides: is there an implication towards Alzheimer's disease and oxidative stress?"
Assay data:1 Active, 3 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Depositor
Esterase Activity Assay from Article 10.3109/14756366.2011.651464: "Analysis of saponins and phenolic compounds as inhibitors of a-carbonic anhydrase isoenzymes."
Assay data:13 Active, 5 Activity ≤ 1 µM, 14 Tested
Esterase Activity Assay from Article 10.3109/14756366.2011.643303: "Carbonic anhydrase inhibitors: in vitro inhibition of a isoforms (hCA I, hCA II, bCA III, hCA IV) by flavonoids."
Assay data:11 Active, 3 Activity ≤ 1 µM, 11 Tested
CA Activity Assay from Article 10.3109/14756366.2011.621122: "Carbonic anhydrase inhibitors: inhibition of human and bovine isoenzymes by benzenesulphonamides, cyclitols and phenolic compounds."
Assay data:10 Active, 4 Activity ≤ 1 µM, 13 Tested
Enzyme Assay from Article 10.3109/14756366.2010.616860: "Polyphenol fatty acid esters as serine protease inhibitors: a quantum-chemical QSAR analysis."
Assay data:9 Active, 25 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on