BioAssay by Target (List) for Gene (Select 11183) - PubChem BioAssay - NCBI

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Select item 19146821.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000753a MAP4K5

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1914682

Summary Related BioAssays by Target

Select item 19135512.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000147b MAP4K5

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1913551

Summary Related BioAssays by Target

Select item 19005293.

Inhibition of MAP4K5 (KHS1) (unknown origin) at 1 uM relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1900529

Summary PubMed Citation Related BioAssays by Target

Select item 18986784.

Inhibition of MAP4K5 (unknown origin) assessed as residual activity at 1 uM by radiometric 33 PanQuinase assay relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1898678

Summary PubMed Citation Related BioAssays by Target

Select item 18951315.

Inhibition of full length C-terminal nanoLuc-tagged human MAP4K5 (KHS1) expressed in HEK293 cells using NanoBRET NanoGlo substrate incubated for 2 hrs in presence of tracer K10 by NanoBRET assay

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1895131

Summary PubMed Citation Related BioAssays by Target

Select item 18951206.

Inhibition of human MAP4K5 (KHS1) by radiometric PanQinase activity assay

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895120

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18951077.

Inhibition of human MAP4K5 (KHS1) at 1 uM by radiometric PanQinase activity assay relative to control (Rvb=50%)

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1895107

Summary PubMed Citation Related BioAssays by Target

Select item 18565848.

Inhibition of MAP4K5 in HEK293 cells by NanoBRET assay

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1856584

Summary PubMed Citation Related BioAssays by Target

Select item 18565659.

Inhibition of human wild type MAP4K5 assessed as remaining activity at 1 uM by MRC screening assay relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1856565

Summary PubMed Citation Related BioAssays by Target

Select item 184935210.

Binding affinity to MAP4K5 (unknown origin) assessed as dissociation constant by competition binding assay

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1849352

Summary Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 183550811.

MAP4K5 DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1835508

Summary Related BioAssays by Target

Select item 183503112.

MAP4K5(h) Kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1835031

Summary Related BioAssays by Target

Select item 183418313.

Inhibition of KHS (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1834183

Summary PubMed Citation Related BioAssays by Target

Select item 179417814.

KinomeScan assay: inhibition of MAP4K5

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Active, 108 Tested

AID:: 1794178

Summary Compounds, Active Related BioAssays by Target

Select item 179372015.

KHS1(M4K5LGY1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793720

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179343116.

KHS1(M4K5LGY1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793431

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179313717.

KHS1(M4K5LGY1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793137

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179273818.

MAP4K5(h) Eurofins kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1792738

Summary Related BioAssays by Target

Select item 179234919.

MAP4K5 ProQinase selectivity panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1792349

Summary Related BioAssays by Target

Select item 179107120.

MAP4K5 (KHS1) Kinase screen

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase kinase 5

Assay data:1 Tested

AID:: 1791071

Summary Related BioAssays by Target

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Target

Proteins (3)
BioAssays with protein sequences specified as targets
RNAi Target, Active (8)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (30)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (6)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (26)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (34)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (40)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (162)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (44)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (1)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (132)
BioAssays extracted from the literature
NIH MLP (2)
BioAssays deposited by the NIH Molecular Libraries Program
Other (71)
BioAssays deposited by other experimentalists

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BioAssay by Target (List) for Gene (Select 11183) (206)
PubChem BioAssay
CLDN14 claudin 14 [Homo sapiens]
CLDN14 claudin 14 [Homo sapiens]
Gene ID:23562

Gene
Gene Links for GEO Profiles (Select 132535595) (1)
Gene
Protein Links for Gene (Select 11183) (34)
Protein
VCPKMT[gene] (29)
ClinVar

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