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Inhibition Assay from US Patent US11325884: "Ketone inhibitors of lysine gingipain"
Assay data:9 Active, 5 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Inhibition of Lysine Gingipain from US Patent US10730826: "Ketone inhibitors of lysine gingipain"
Assay data:59 Active, 39 Activity ≤ 1 nM, 66 Activity ≤ 1 µM, 66 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Cathepsin H (h) Eurofins-Cerep enzyme and uptake assay
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of cathepsin H (unknown origin) at 10 uM
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Inhibition of Cathepsin H (unknown origin) at 10 uM
Reversible competitive inhibition of human cathepsin H using fluorogenic AMC-derived peptide substrate assessed as reduction in residual activity preincubated for 30 mins followed by substrate addition
Assay data:2 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of human cathepsin H using fluorogenic AMC-derived peptide substrate assessed as reduction in residual activity preincubated for 30 mins followed by substrate addition
Assay data:1 Active, 4 Tested
Competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-inhibitor complex using R-AMC as substrate in presence of pH 6 phosphate buffer by fluorescence assay
Non-competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-substrate-inhibitor complex using R-AMC as substrate in presence of pH 6 phosphate buffer by fluorescence assay
Assay data:2 Tested
Non-competitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-inhibitor complex using R-AMC as substrate in presence of pH 6 phosphate buffer by fluorescence assay
Uncompetitive inhibition of human liver cathepsin H assessed as inhibitory constant for enzyme-substrate-inhibitor complex using R-AMC as substrate in presence of pH 6 phosphate buffer by fluorescence assay
Human cathepsin H (C1: Papain)
Assay data:2 Active, 2 Tested
Inhibition of human recombinant cathepsin H
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced TNF-alpha response in human macrophages_Primary screen TNF readout
Assay data:2853 Active, 18113 Tested
SummaryRelated BioAssays by Same Project
Inhibition of Cathepsin H (unknown origin) at 0.25 x 10'-4 M
Inhibition of Cathepsin H (unknown origin) at 1 x 10'-4 M
Inhibition of human liver cathepsin H
Assay data:1 Active, 1 Tested
A screen to identify synthetic lethal interactions with E-cadherin in an MCF10A isogenic cell line
Assay data:2442 Active, 18052 Tested
SummaryPubMed Citation
A screen to identify genes that regulate lymphatic endothelial cell migration - Primary Screen
Assay data:1034 Active, 18120 Tested
SummaryRelated BioAssays by Depositor
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