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Displacement of [3H]NT from human NTS2 receptor expressed in HEK293 cells
Assay data:35 Active, 2 Activity ≤ 1 nM, 32 Activity ≤ 1 µM, 35 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]NT(8 to 13) from human NTS2 receptor expressed in HEK293 cells
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
Agonist activity at NTR2 (unknown origin) expressed in human U2OS cells coexpressing beta-arrestin by GFP reporter gene assay
Assay data:45 Tested
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity to NTR2 (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
RNAi screen for vorinostat resistance genes - Primary Screen
Assay data:450 Active, 18118 Tested
SummaryPubMed Citation
Druggable Genome siRNA Screen for Enhancers of Camptothecin in MDA-MB-231 Breast Cancer Cells
Assay data:167 Active, 26449 Tested
Summary
Genome-wide high-content siRNA screens for regulators of Parkin translocation in selective mitophagy (Ambion Library)
Assay data:9227 Active, 64752 Tested
Genome-wide high-content siRNA screens for regulators of Parkin translocation in selective mitophagy (Dharmacon Library)
Assay data:826 Active, 18119 Tested
An siRNA screen for human genes that are involved in human papilloma virus (HPV) E2 transcriptional repression of the E6 and E7 oncogenes
Assay data:497 Active, 21019 Tested
SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2
Assay data:20 Active, 87 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activity at 3 uM in presence of SR142948A
Assay data:1 Tested
Ratio of compound EC50 to neurotensin EC50 for human NTS2 receptor
Assay data:4 Tested
Agonist activity at human NTS2 receptor expressed in HEK293 cells assessed as inhibition of constitutive activity on MAPK-mediated luciferase activity
Assay data:5 Active, 5 Activity ≤ 1 µM, 5 Tested
Agonist activity at NTR2 in human U2OS cells after 1 hr by beta-arrestin GFP reporter gene assay
Assay data:2 Tested
SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay
Assay data:13 Active, 122 Tested
Binding affinity to human NTR2 by gamma counting
Displacement of [125I]Tyr3NT from human NTS2 receptor expressed in COS7 cells
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Binding affinity at human NTS2 receptor
Evaluated for binding affinity by inhibiting binding of [125I]Tyr(3)-NT to human Neurotensin receptor 2
Assay data:21 Active, 6 Activity ≤ 1 nM, 21 Activity ≤ 1 µM, 21 Tested
Binding ability to compete with [125I]Tyr3-NT (0.15 nM) for human NT receptors cloned in CHO cells.
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
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