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Glutamate, Kainate Eurofins Panlabs panel
Assay data:1 Tested
SummaryRelated BioAssays by Target
Glutamate, Non-Selective Eurofins-Panlabs radioligand binding assay
Glutamate, Kainate Eurofins-Panlabs radioligand binding assay
Assay data:5 Tested
Displacement of [3H]kainic acid from rat Glutamate receptor, ionotropic kainate at 10 uM after 60 mins by scintillation counting method relative to control
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of rat brain Glutamate receptor, ionotropic kainate assessed as [3H]kainic acid uptake at 10 uM after 60 mins by scintillation counting analysis relative to control
Activity at rat recombinant GluK2/GluK5 receptor expressed in Xenopus oocytes assessed as effect on glutamate-induced response at 3 uM by two-electrode voltage clamp technique relative to control
Late-stage radioligand binding dose response assay to identify inhibitors of NADPH oxidase 1 (NOX1): PDSP screen Ki
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Binding affinity to rat cloned KA2 receptor
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]kainic acid from kainate receptor at 0.5 uM
Antagonist activity against rat KA receptor assessed by inhibition of kainate-induced membrane current at 1 uM
Antagonist activity against rat KA receptor assessed by inhibition of kainate-induced membrane current at 100 uM
Assay data:4 Tested
Agonist activity at rat KA receptor assessed by generation of membrane current at 100 uM relative to control in presence of 10 uM cyclothiazide
Agonist activity at rat KA receptor assessed by generation of membrane current at 100 uM relative to control
Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibers at 100 uM
Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibers
Assay data:8 Active, 2 Activity ≤ 1 µM, 14 Tested
Displacement of [3H]KAIN from kainate receptor in rat brain
In vitro inhibitory concentration against KA receptor using [3H]KA
Assay data:8 Tested
Displacement of [3H]KA from glutamate receptor of rat brain synaptosomes
Assay data:10 Tested
Compound was tested for inhibition of [3H]kainate (KA) binding to cortical membranes
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Binding affinity towards kainate receptor to rat cortical membrane using [3H]kainate as radioligand
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