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In vitro binding ability against Luteinizing hormone-releasing hormone release in rat pituitary cells; ND denotes not determined
Assay data:2 Tested
SummaryPubMed CitationRelated BioAssays by Target
In vivo luteinizing hormone inhibiting potency in rats is expressed as negative logarithm of the concentration (antagonist)
Assay data:4 Active, 2 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
In vivo inhibition of leutenising hormone in rats.
Assay data:21 Active, 1 Activity ≤ 1 nM, 21 Activity ≤ 1 µM, 21 Tested
In vivo luteinizing hormone releasing potency in rats is expressed as negative logarithm of the concentration of compound (agonist)
Assay data:1 Tested
Leutinising hormone releasing potency in rats is expressed as negative logarithm of the concentration of agonist
Leutinising hormone releasing potency in rats is expressed as negative logarithm of the concentration of compound (agonist)
Compounds were tested for the effective dose to induce luteinizing hormone (LH) release in rat pituitary receptors
Compound was evaluated for its antagonism in rat primary pituitary cell assay (rLH): NA=Data not available
Negative logarithm of equilibrium dissociation constant in the rat pituitary Luteinizing Hormone Releasing Hormone (LHRH) receptor binding assay
Assay data:2 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assay
Assay data:10 Active, 7 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
Luteinizing hormone inhibiting potency in rats is expressed as negative logarithm of the concentration (antagonist)
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
In vitro binding affinity towards Luteinizing hormone receptor from rat pituitary cells is expressed as negative logarithm of the equilibrium dissociation constant
Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested
In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilibrium dissociation constant
Assay data:33 Active, 4 Activity ≤ 1 nM, 31 Activity ≤ 1 µM, 33 Tested
In vitro binding ability against Luteinizing hormone-releasing hormone release in rat pituitary cells
Assay data:4 Active, 2 Activity ≤ 1 nM, 4 Activity ≤ 1 µM, 4 Tested
Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-induced cAMP production preincubated for 30 mins followed by agonist solution addition after 30 mins by cell based TR-FRET assay
Assay data:5 Active, 4 Activity ≤ 1 µM, 5 Tested
Antiovulatory activity in Sprague-Dawley rats expressed as the percentage rats blocked at a dose 3 microg
Assay data:13 Tested
In vitro histamine-release activity by using peritoneal cells from male Sprague-Dawley rats in a standard assay
Assay data:19 Tested
Efficacy at LH receptor in Sprague-Dawley rat Leydig cells assessed as production of testosterone after 3 hrs
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Agonist activity at LH-RH receptor in rat pituitary gland assessed as change in luteinizing hormone secretion at 100000 ng/ml
Assay data:4 Tested
Agonist activity at LH-RH receptor in rat pituitary gland assessed as change in FSH secretion at 100000 ng/ml
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