Warning: The NCBI web site requires JavaScript to function. more...
An official website of the United States government
The .gov means it's official. Federal government websites often end in .gov or .mil. Before sharing sensitive information, make sure you're on a federal government site.
The site is secure. The https:// ensures that you are connecting to the official website and that any information you provide is encrypted and transmitted securely.
Antagonist activity at human neuropeptide Y2 receptor
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to Neuropeptide Y Y2 receptor at 10 uM by radioligand binding assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Displacement of [125I]peptide YY from human recombinant Y2 receptor expressed in KAN-TS cells
Antagonist activity at human NPY Y2 receptor in KAN-TS cells by [35]GTPgammaS assay
Assay data:29 Active, 27 Activity ≤ 1 µM, 29 Tested
Displacement of [125I]-Peptide YY from neuropeptide Y2 receptor at 1 to 3 uM
Displacement of [125I]peptide YY from NPY2 receptor in human KAN-TS cells
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity to human recombinant neuropeptide Y2 receptor
Antagonist activity at human NPY Y2 receptor expressed in HEK293 cells assessed as inhibition of calcium level by FLIPR assay
Displacement of [125I]pig PPY from human NPY2 receptor expressed in CHOK1 cells by scintillation counting
Assay data:2 Tested
Displacement of [125I]peptideYY from neuropeptide Y2 receptor in human KAN-TS cells at 10 uM after 60 mins by scintillation counting
Displacement of [125I]PYY from human neuropeptide Y2 receptor expressed in human SK-N-BE2 cells after 40 mins
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
Inhibition of human NPY Y2 receptor
Displacement of [125I]-PYY from human NPYY2 receptor
Antagonist activity at human neuropeptide Y2 receptor expressed in HEK293 cells by [35S]GTPgammaS binding assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Binding affinity to human NPY Y2 receptor
Antagonist activity at human neuropeptide Y2 receptor by [35]GTPgammaS assay
Binding affinity to neuropeptide Y2 receptor
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assay
Assay data:27 Active, 23 Activity ≤ 1 µM, 28 Tested
Binding affinity to human neuropeptide Y2 receptor
Filters: Manage Filters
Your browsing activity is empty.
Activity recording is turned off.
Turn recording back on