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Inhibition of PI3K-P85 phosphorylation in human HT-29 cells at 4 uM incubated for 72 hrs by Western blot analysis
Assay data:1 Active, 1 Tested
SummaryRelated BioAssays by Target
Inhibition of PI3K-P85 phosphorylation in human HT-29 cells at 2 uM incubated for 72 hrs by Western blot analysis
Inhibition of PI3K-P85 phosphorylation in human HT-29 cells at 1 uM incubated for 72 hrs by Western blot analysis
Inhibition of recombinant PI3K p110alpha/p85 (unknown origin) incubated for 1 hr in presence of gamma[33P]ATP by scintillation counting analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of human P13Kalpha
Inhibition of PI3 kinase p110alpha/p85alpha (unknown origin) at 1 uM relative to control
Assay data:1 Tested
Inhibition of PI3 Kinase p110delta/p85alpha (unknown origin) at 1 uM relative to control
Inhibition of P13 kinase p110beta/p85alpha (unknown origin) at 1 uM relative to control
Assay of ATR Kinase Activity from US Patent US20230271968: "PYRAZOLOPYRIMIDINE COMPOUND USED AS ATR KINASE INHIBITOR"
Assay data:24 Active, 24 Activity ≤ 1 µM, 24 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of PI3K p110alpha/p85alpha (unknown origin) using PIP2 as substrate preincubated for 15 mins followed by substrate addition measured after 1 hr in presence of ATP by TR-FRET assay
Assay data:6 Active, 6 Activity ≤ 1 µM, 6 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of p110alpha/p85alpha (unknown origin) at 50 nM by Z'LYTE screening method relative to control
Assay data:12 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of recombinant human full length PI3K p110delta/p85a using phosphatidylinositol-4, 5-bisphosphate as substrate incubated for 40 mins in presence of [gamma33P]ATP by radiometric scintillation counting analysis
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Radioisotope Filter Binding Assay from US Patent US10844038: "1,2-dithiolane compounds useful in neuroprotection, autoimmune and cancer diseases and conditions"
Assay data:12 Active, 9 Activity ≤ 1 µM, 12 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
PI3K (p110delta/p85alpha) (h) [Non-Radioactive Assay] from US Patent US10751339: "Substituted aminopyrimidine compounds and methods of use"
Assay data:13 Active, 13 Activity ≤ 1 µM, 13 Tested
PI3K (p110beta/p85alpha) (h) [Non-Radioactive Assay] from US Patent US10751339: "Substituted aminopyrimidine compounds and methods of use"
Assay data:11 Active, 9 Activity ≤ 1 µM, 13 Tested
PI3K (p110alpha/p85alpha) (h) [Non-Radioactive Assay] from US Patent US10751339: "Substituted aminopyrimidine compounds and methods of use"
Assay data:9 Active, 4 Activity ≤ 1 µM, 13 Tested
Fluorescent Determination of PI3K Enzyme Activity from US Patent US10611777: "Imidazopyridazine compounds and their use"
Assay data:69 Active, 8 Activity ≤ 1 nM, 69 Activity ≤ 1 µM, 69 Tested
PI3K p110delta/p85alpha (Human), Non-radioactive Assay from US Patent US10457677: "Imidazolonylquinolines and the use thereof as ATM kinase inhibitors"
Assay data:57 Tested
SummaryRelated BioAssays by DepositorRelated BioAssays by Target
PI3K p110beta/p85alpha (Human), Non-radioactive Assay from US Patent US10457677: "Imidazolonylquinolines and the use thereof as ATM kinase inhibitors"
Assay data:50 Tested
PI3K p110alpha/p85alpha (Human), Non-radioactive Assay from US Patent US10457677: "Imidazolonylquinolines and the use thereof as ATM kinase inhibitors"
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