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Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24 to 48 hrs by luciferase reporter gene assay relative to control
Assay data:24 Tested
SummaryRelated BioAssays by Target
Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24 to 48 hrs by luciferase reporter gene assay
Assay data:24 Active, 24 Activity ≤ 1 µM, 24 Tested
Agonist activity at human PPAR-delta assessed as receptor transactivation by measuring maximum induction of alkaline phosphatase activity
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Agonist activity at PPARdelta (unknown origin)
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Agonist activity at human PPARdelta
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Activation of PPARdelta (unknown origin) at 10 uM
Assay data:1 Tested
Binding affinity to PPARdelta (unknown origin) upto 10 uM by TR-FRET-based competitive binding assay
Assay data:11 Tested
Agonist activity at human PPARdelta at 0.0075 uM incubated for 22 to 24 hrs by luciferase assay relative to control
Agonist activity at human PPARdelta at 0.013 to 100 uM incubated for 22 to 24 hrs by luciferase assay relative to GW0742
Assay data:5 Tested
Agonist activity at human PPARdelta at 17 uM incubated for 22 to 24 hrs by luciferase assay relative to GW0742
Displacement of Fluormone Pan-PPAR Green from GST-tagged human PPAR-delta ligand binding domain at 10 uM by LanthaScreen TR-FRET competitive binding assay
Assay data:12 Tested
Binding affinity to PPARdelta (unknown origin)
Assay data:1 Active, 1 Tested
Agonist activity at PPARdelta (unknown origin) relative to control
Agonist activity at PPARdelta (unknown origin) at 20 uM relative to control
Assay data:1 Active, 1 Activity ≤ 1 µM, 4 Tested
Inverse agonist activity at human PPARdelta expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression by measuring maximum efficacy preincubated for 6 hrs followed by luciferin addition by luminescence method
Assay data:2 Tested
Inverse agonist activity at human PPARdelta expressed in CHO cells co-expressing GAL4-NHR-LBD assessed as transcriptional repression preincubated for 6 hrs followed by luciferin addition by luminescence method
Assay data:1 Active, 5 Tested
Agonist activity at human PPARdelta expressed in HEK293T cells incubated for 12 to 14 hrs by Dual-Glo luciferase assay
Assay data:3 Active, 1 Activity ≤ 1 µM, 4 Tested
Displacement of fluormone pan-PPARgreen from GST-tagged human PPARdelta ligand binding domain at 10 uM by LanthaScreen TR-FRET competitive binding assay
Partial agonist activity at PPARdelta (unknown origin) assessed as increase in fluorescein labeled PRIP/RAP250 coactivator peptide requirement by Lanthascreen TR-FRET assay
Assay data:1 Active, 1 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
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