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Inhibition of human recombinant Enteropeptidase assessed as inhibition based on initial velocity using 5FAM-Abu-Gly-Asp -Asp-Asp -Lys-Ile-Val-Gly-Gly-Lys-(CPQ2)-Lys-Lys-NH2 as substrate by fluorescence based plate reader method
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity human recombinant Enteropeptidase assessed as dissociation of half life using FAM-Abu-Gly-Asp -Asp-Asp-Lys-Ile -Val-Gly-Gly-Lys-(CPQ2)-Lys -Lys-NH2 as substrate preincubated for 2 hrs followed by substrate addition by rapid dilution assay
Assay data:4 Tested
Inhibition of human recombinant Enteropeptidase assessed as inhibition based on steady state using 5FAM-Abu-Gly-Asp -Asp-Asp -Lys-Ile-Val-Gly-Gly-Lys-(CPQ2)-Lys-Lys-NH2 as substrate incubated for 120 mins by fluorescence based plate reader method
Assay data:17 Active, 2 Activity ≤ 1 nM, 17 Activity ≤ 1 µM, 17 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human recombinant Enteropeptidase assessed as inhibition based on initial velocity using 5FAM-Abu-Gly-Asp -Asp-Asp -Lys-Ile-Val-Gly-Gly-Lys-(CPQ2)-Lys-Lys-NH2 as substrate incubated for 6 mins by fluorescence based plate reader method
Assay data:16 Active, 14 Activity ≤ 1 µM, 17 Tested
Enteropeptidase Inhibition Assay from US Patent US11447480: "Compound exhibiting enteropeptidase inhibitory activity"
Assay data:83 Active, 14 Activity ≤ 1 nM, 83 Activity ≤ 1 µM, 83 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition Assay from US Patent US9346821: "Heterocyclic carboxylic acid ester derivative"
Assay data:33 Active, 32 Activity ≤ 1 nM, 33 Activity ≤ 1 µM, 33 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Enteropeptidase Inhibition Assay from US Patent US9227949: "Heteroarylcarboxylic acid ester derivative"
Assay data:94 Active, 53 Activity ≤ 1 nM, 94 Activity ≤ 1 µM, 94 Tested
Inhibition Assay from US Patent US9024044: "Heteroarylcarboxylic acid ester derivative"
Assay data:81 Active, 42 Activity ≤ 1 nM, 81 Activity ≤ 1 µM, 81 Tested
Inhibition Assay from US Patent US8609715: "Heteroarylcarboxylic acid ester derivative"
Assay data:129 Active, 72 Activity ≤ 1 nM, 129 Activity ≤ 1 µM, 129 Tested
Inhibitory Activity Assay from US Patent US9655879: "Heteroarylcarboxylic acid ester derivative"
Inhibition of full length recombinant human EP expressed in CHO cells assessed as ratio of Kinact/Kiapp
Assay data:7 Tested
Inhibition of full length recombinant human EP expressed in CHO cells assessed as protease activity using 2-naphthylamine as substrate at 10 uM by fluorescence assay relative to control
Assay data:44 Tested
Inhibition of full length recombinant human EP expressed in CHO cells assessed as protease activity using 2-naphthylamine as substrate at 1 uM by fluorescence assay relative to control
Inhibition of full length recombinant human EP expressed in CHO cells assessed as protease activity using 2-naphthylamine as substrate at 0.1 uM by fluorescence assay relative to control
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced TNF-alpha response in human macrophages_Primary screen TNF readout
Assay data:2853 Active, 18113 Tested
SummaryRelated BioAssays by Same Project
A screen to identify synthetic lethal interactions with E-cadherin in an MCF10A isogenic cell line
Assay data:2442 Active, 18052 Tested
SummaryPubMed Citation
A screen to identify genes that regulate lymphatic endothelial cell migration - Primary Screen
Assay data:1034 Active, 18120 Tested
SummaryRelated BioAssays by Depositor
Identification of proteins required for the processing of the EWS-FLI1 nascent transcript
Assay data:59220 Tested
InfectX: Pathogen infection siRNA screens
Assay data:115372 Tested
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