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Millipore: Percentage of residual kinase activity of PAK7 at 1uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA
Assay data:158 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of PAK5 (unknown origin) at 0.1 uM
Assay data:1 Tested
Inhibition of PAK5 (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human PAK5 assessed as residual activity at 1 uM relative to control
Competitive binding affinity to PAK7/PAK5 (unknown origin) at 10 uM in presence of ATP relative to control
Assay data:6 Tested
Inhibition of PAK7 (unknown origin) at 10 uM relative to control
RNAi screen for vorinostat resistance genes - Primary Screen
Assay data:450 Active, 18118 Tested
SummaryPubMed Citation
Druggable Genome siRNA Screen for Enhancers of Camptothecin in MDA-MB-231 Breast Cancer Cells
Assay data:167 Active, 26449 Tested
Summary
Inhibition of PAK7 (unknown origin) assessed as remaining activity at 1 uM relative to control
Inhibition of PAK5 (unknown origin) using [gamma-33P]ATP assessed as residual activity at 3 uM
Inhibition of PAK7 (unknown origin) assessed as remaining activity at 10 uM relative to control
Assay data:2 Tested
AT1R-EGFR transactivation kinome screen - primary
Assay data:50 Active, 714 Tested
Millipore: Percentage of residual kinase activity of PAK7 at 10uM relative to control. Control inhibitor: Staurosporine at 10.0uM. Buffer: 8 mM MOPS pH 7.0, 0.2 mM EDTA
Assay data:3 Tested
Inhibition of PAK5 assessed as residual activity at 10 uM
Inhibition of PAK5 assessed as residual activity at 1 uM
Inhibition of PAK7 assessed as residual activity at 10 uM relative to control
Inhibition of PAK7 at 1 uM
Inhibition of PAK5 assessed as residual activity at 1 uM relative to control
Inhibition of PAK5 assessed as residual activity at 10 uM relative to control
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