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RNAi screen for vorinostat resistance genes - Primary Screen
Assay data:450 Active, 18118 Tested
SummaryPubMed Citation
Inhibition of acid-induced matriptase activation in human HaCaT cells using mAb M24 after 30 mins by Western blot analysis
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of acid-induced matriptase activation in human HaCaT cells using mAb M69 after 30 mins by Western blot analysis
Inhibition of acid-induced matriptase-mediated prostasin activation in human HaCaT cells assessed as decrease in prostatin-HAI-1 complex after 30 mins by Western blot analysis
Inhibition of acid-induced matriptase activation in human 184A1N4 cells assessed as enzyme-HAI-1 complex using mAb M24 at 5 uM after 30 mins by Western blotting
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Genome-wide high-content siRNA screens for regulators of Parkin translocation in selective mitophagy (Dharmacon Library)
Assay data:826 Active, 18119 Tested
Genome-wide high-content siRNA screens for regulators of Parkin translocation in selective mitophagy (Ambion Library)
Assay data:9227 Active, 64752 Tested
Inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate at 2.5 nM by fluorimetric analysis
Irreversible inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 20 mins prior to substrate addition measured for 75 mins by fluorimetric analysis
Reversible inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 20 mins prior to substrate addition measured for 75 mins by fluorimetric analysis
Tight binding inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate incubated for 15 mins prior to substrate addition measured for 30 mins by fluorimetric analysis
Assay data:5 Active, 2 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Mixed inhibition of human matriptase expressed in Drosophila melanogaster S2 cells using Boc-QAR-AMC as substrate by fluorimetric analysis
Assay data:2 Active, 1 Activity ≤ 1 µM, 2 Tested
Druggable Genome siRNA Screen for Enhancers of Camptothecin in MDA-MB-231 Breast Cancer Cells
Assay data:167 Active, 26449 Tested
Summary
Inhibition of acid-induced matriptase activation in human 184A1N4 cell homogenate using mAb M69 after 30 mins by Western blot analysis
Assay data:4 Tested
Binding affinity to human matriptase assessed as half life of deacylated enzyme
Assay data:2 Tested
Inhibition of human matriptase measured after 15 mins at pH 8 by fluorescence assay
Assay data:2 Active, 2 Activity ≤ 1 µM, 7 Tested
Inhibition of matriptase-SP1 (615 to 855) (unknown origin) expressed in Escherichia coli BL21(DE3) using Boc-Gln-Ala-Arg-7-amido-4-methyl coumarin hydrobromide as substrate by fluorescence assay
Assay data:13 Active, 10 Activity ≤ 1 µM, 14 Tested
Reversible inhibition of matriptase (unknown origin) using Boc-Gln-Ala-Arg-AMC as substrate after 15 to 60 mins by fluorescence assay
Assay data:16 Active, 16 Tested
Inhibition of matriptase (unknown origin) using Boc-Gln-Ala-Arg-AMC as substrate at 50 uM after 15 mins by fluorescence assay
Assay data:9 Tested
Inhibition of matriptase (unknown origin) using Boc-Gln-Ala-Arg-AMC as substrate after 15 mins by fluorescence assay
Assay data:7 Tested
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