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Selectivity interaction (KinomeScan (DiscoverX)) EUB0000307b DDR1
Assay data:1 Tested
SummaryRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000710a DDR1
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000703a DDR1
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000703a DDR1
Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000703a DDR1
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000312b DDR1
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000312b DDR1
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000132b DDR1
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000132b DDR1
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000147b DDR1
Affinity Biochemical interaction (Radiometric assay (10 M ATP, Reaction Biology)) EUB0000156b DDR1
Affinity Biochemical interaction (Radiometric assay (10 M ATP, Reaction Biology)) EUB0000005b DDR1
Affinity Biochemical interaction (KdELECT (DiscoverX)) EUB0000713a DDR1
Assay data:1 Active, 1 Activity ≤ 1 nM, 1 Activity ≤ 1 µM, 1 Tested
Affinity Biochemical interaction (Enzyme kinetic assay (Reaction Biology)) EUB0000712a DDR1
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000156b DDR1
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000005b DDR1
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000713a DDR1
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000712a DDR1
Affinity On-target Cellular interaction (NanoBRET assay (HEK293T cells)) EUB0000703a DDR1
Inhibition of human DDR1 at 100 nM by KINOMEscan assay relative to control
SummaryPubMed CitationRelated BioAssays by Target
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