BioAssay by Target (List) for Gene (Select 80122) - PubChem BioAssay - NCBI

Warning: The NCBI web site requires JavaScript to function. more...

Links from Gene

Items: 1 to 20 of 127

<< First< Prev

Page of 7

Select item 19527671.

Inhibition of wild type human YSK4 in presence of ATP by radiometric kinase assay

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1952767

Summary PubMed Citation Related BioAssays by Target

Select item 19527532.

Inhibition of wild type human YSK4 at 1 uM by DiscoverX scanMAX assay relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1952753

Summary PubMed Citation Related BioAssays by Target

Select item 19488853.

Inhibition of YSK4 (unknown origin) assessed as dissociation constant

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1948885

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19488824.

Inhibition of YSK4 (unknown origin) at 1 uM relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:3 Tested

AID:: 1948882

Summary PubMed Citation Related BioAssays by Target

Select item 19193475.

In Vitro Effect Assay from US Patent US11608319: "Beta-amino acid derivative, kinase inhibitor and pharmaceutical composition containing the same, and method for performing an in vivo related application that benefits from the inhibition of a kinase"

Source:: BindingDB

Protein Targets:: Mitogen-activated protein kinase kinase kinase 19; ...
Total:: 1

Assay data:7 Activity ≤ 1 µM, 15 Tested

AID:: 1919347

Summary Compounds, activity ≤ 1 µM Related BioAssays by Depositor Related BioAssays by Target

Select item 19154366.

Selectivity interaction (Kinase Panel (competition binding assay)) EUB0000589aTFA MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1915436

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 19140797.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000138c MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1914079

Summary Related BioAssays by Target

Select item 19139588.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000702a MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1913958

Summary Related BioAssays by Target

Select item 19139329.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000701a MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1913932

Summary Related BioAssays by Target

Select item 191390710.

Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000305b MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1913907

Summary Related BioAssays by Target

Select item 191390611.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000305b MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1913906

Summary Related BioAssays by Target

Select item 191390512.

Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000305b MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913905

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 189355913.

Inhibition of wild-type human partial length YSK4 (T1019 to H1328 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1893559

Summary PubMed Citation Related BioAssays by Target

Select item 185655414.

Inhibition of wild-type human partial length YSK4 (T1019 to H1328 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1856554

Summary PubMed Citation Related BioAssays by Target

Select item 183564115.

YSK4 DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1835641

Summary Related BioAssays by Target

Select item 183437716.

Inhibition of YSK4 (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1834377

Summary PubMed Citation Related BioAssays by Target

Select item 182346617.

Inhibition of YSK4 (unknown origin) at 1 uM by kinome scan method

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Active, 1 Tested

AID:: 1823466

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 180725618.

Inhibition of wild-type human partial length YSK4 (T1019 to H1328 residues) expressed in mammalian expression system at 1 uM by Kinomescan method

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Active, 1 Tested

AID:: 1807256

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 179440019.

KinomeScan assay: inhibition of YSK4

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:4 Active, 108 Tested

AID:: 1794400

Summary Compounds, Active Related BioAssays by Target

Select item 179256620.

NanoBRET with MAP3K19

Source:: ChEMBL

Protein Target:: Mitogen-activated protein kinase kinase kinase 19

Assay data:1 Tested

AID:: 1792566

Summary Related BioAssays by Target

<< First< Prev

Page of 7

Supplemental Content

Filters: Manage Filters

Refine your results

• What's this?

Target

Proteins (1)
BioAssays with protein sequences specified as targets
RNAi Target, Active (8)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (23)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (2)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (17)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (2)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (22)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (40)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (82)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (45)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (2)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (66)
BioAssays extracted from the literature
NIH MLP (1)
BioAssays deposited by the NIH Molecular Libraries Program
Other (59)
BioAssays deposited by other experimentalists

Actions on your results

View or Download BioAssay in PubChem

Find related data

Recent activity

Clear Turn Off Turn On

BioAssay by Target (List) for Gene (Select 80122) (127)
PubChem BioAssay

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...

You are here: NCBI > Chemicals & Bioassays > PubChem BioAssay