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CAMK2D SGC Tm panel (DSF)
Assay data:1 Tested
SummaryRelated BioAssays by Target
Thermal Shift Assay. Domain: start/stop: T11-N335
Assay data:27 Tested
CAMK2D DiscoveRx kinase panel
CaMKIIdelta(h) Kinase panel
Inhibition of CAMK2D (unknown origin) at 1 uM
SummaryPubMed CitationRelated BioAssays by Target
Inhibition Assay from US Patent US10759792: "CaMKII inhibitors and uses thereof"
Assay data:16 Active, 26 Activity ≤ 1 µM, 26 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
In Vitro Inhibition Assay from US Patent US8975250: "5 oxo-5,8-dihydropyrido[2,3-d]pyrimidine derivatives as CaMKII kinase inhibitors for treating cardiovascular diseases"
Assay data:13 Active, 13 Activity ≤ 1 µM, 13 Tested
CaMKII Cell-Based Activity from US Patent US10100058: "Fused heterocyclic compounds as CaM kinase inhibitors"
Assay data:348 Active, 345 Activity ≤ 1 µM, 349 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
CaMKII delta Biochemical Assay from US Patent US10100058: "Fused heterocyclic compounds as CaM kinase inhibitors"
Assay data:364 Active, 177 Activity ≤ 1 nM, 364 Activity ≤ 1 µM, 364 Tested
KinomeScan assay: inhibition of CAMK2D
Assay data:108 Tested
CaMK2delta(CA2DCGT1) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
CaMKIIdelta(h) Eurofins kinase panel
CAMK2D ProQinase selectivity panel
CAMK2D (CaMKII delta) Kinase screen
CAMK2D Invitrogen selectivity data (BI)
CaMKIIdelta (h) Eurofins Kinase panel
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