BioAssay by Target (List) for Gene (Select 83810) - PubChem BioAssay - NCBI

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Select item 2700251.

Antagonist activity against rat TRPV1 assessed as inhibition of capsaicin-induced calcium influx by FLIPR assay

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Tested

AID:: 270025

Summary PubMed Citation Related BioAssays by Target

Select item 2650722.

Decrease in carrageenan-induced thermal hyperalgesia in rat at 30 mg/kg, po

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Tested

AID:: 265072

Summary PubMed Citation Related BioAssays by Target

Select item 2650733.

Activity against capsaicin-induced intracellular calcium ion increase in CHO cells expressing rat TRPV1 assessed by patch clamp

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 265073

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 2650744.

Activity at rat TRPV1 as inhibition of capsaicin-induced intracellular calcium ion increase in CHO cells

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 265074

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 2654805.

Antagonist activity against capsaicin-mediated activation of rat TRPV1 by FLIPR

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:21 Tested

AID:: 265480

Summary PubMed Citation Related BioAssays by Target

Select item 2655046.

Activity against capsaicin-induced secondary hyperalgesia assessed as reversal of allodynia in rat at 10 mg/kg, po after 2 hrs

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Active, 1 Tested

AID:: 265504

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 2655057.

Activity against capsaicin-induced secondary hyperalgesia assessed as reversal of allodynia in rat at 30 mg/kg, po after 2 hrs

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Active, 1 Tested

AID:: 265505

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 2663148.

Antagonist activity against capsaicin-induced 45calcium ion uptake in CHO cells expressing rat TRPV1

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:77 Active, 4 Activity ≤ 1 nM, 58 Activity ≤ 1 µM, 83 Tested

AID:: 266314

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 2663159.

Antagonist activity against acid-induced 45calcium ion uptake in CHO cells expressing rat TRPV1 at pH5

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:68 Active, 6 Activity ≤ 1 nM, 61 Activity ≤ 1 µM, 83 Tested

AID:: 266315

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 26632210.

Antinociceptive activity in po dosed Sprague-Dawley rat assessed as ability to block capsaicin-induced paw flinching

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Tested

AID:: 266322

Summary PubMed Citation Related BioAssays by Target

Select item 26632311.

Antinociceptive activity in Sprague-Dawley rat assessed as reversal of CFA-induced thermal hyperalgesia

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Active, 1 Tested

AID:: 266323

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 27002312.

Antagonist activity against rat TRPV1 assessed as inhibition of acid-induced calcium influx by FLIPR assay

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 270023

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 25767913.

Effect on neuropathic mechanical hyperalgesia in rat at 1 hr

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:1 Tested

AID:: 257679

Summary PubMed Citation Related BioAssays by Target

Select item 27133214.

Antagonist activity against low pH(5.0-5.5)-activated rat VR1

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:54 Active, 2 Activity ≤ 1 nM, 49 Activity ≤ 1 µM, 64 Tested

AID:: 271332

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 28934915.

Displacement of [3H]RTX from rat TRPV1 receptor expressed in CHO cells

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:19 Active, 13 Activity ≤ 1 µM, 20 Tested

AID:: 289349

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 28935016.

Agonist activity at rat TRPV1 receptor expressed in CHO cells by Ca2+ uptake assay

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:20 Tested

AID:: 289350

Summary PubMed Citation Related BioAssays by Target

Select item 28935117.

Antagonist activity at rat TRPV1 receptor expressed in CHO cells by Ca2+ uptake assay

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:18 Active, 16 Activity ≤ 1 µM, 20 Tested

AID:: 289351

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 29195118.

Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium influx

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:13 Active, 12 Activity ≤ 1 µM, 23 Tested

AID:: 291951

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 29195219.

Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of acid-induced calcium influx

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:9 Active, 6 Activity ≤ 1 µM, 23 Tested

AID:: 291952

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 29196920.

Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-induced calcium influx

Source:: ChEMBL

Protein Target:: Transient receptor potential cation channel subfamily V member 1

Assay data:19 Active, 2 Activity ≤ 1 nM, 16 Activity ≤ 1 µM, 29 Tested

AID:: 291969

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

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Target

Proteins (1)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (208)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (48)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (163)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (185)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (378)
BioAssays extracted from the literature

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BioAssay by Target (List) for Gene (Select 83810) (378)
PubChem BioAssay
Taxonomy Links for Protein (Select 557700751) (1)
Taxonomy
PubChem Compound Links for Gene (Select 798361) (2)
PubChem Compound
Gene Links for GEO Profiles (Select 12582484) (1)
Gene
CAPN7 calpain 7 [Homo sapiens]
CAPN7 calpain 7 [Homo sapiens]
Gene ID:23473

Gene

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