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Binding affinity towards human CCKBR in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:6 Active, 1 Activity ≤ 1 µM, 856 Tested
SummaryRelated BioAssays by Target
Binding affinity to human CCK2R expressed in human A-431 cells
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Selectivity interaction (CEREP Wide Ligand screening panel (ion channels, receptors, enzymes)) EUB0000304b CCKBR
Assay data:1 Tested
Agonist activity at human CCK2R expressed in HEK293 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by AlphaScreen assay
Assay data:1 Active, 8 Activity ≤ 1 µM, 10 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Antagonist activity at pig cerebral cortex CCK2 human by Packbard-Cobra counter analysis
Cholecystokinin CCK2 (CCKB) Eurofins-Panlabs radioligand binding assay
CCKB/H Eurofins SafetyScreen44 (BI)
Radioligand Labeled Binding Assay and Phosphatidylinositol Hydrolysis Assay for the CCK Receptor from Article 10.1021/jm050921q: "Structure-activity relationships of bifunctional peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors."
Assay data:16 Active, 1 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 16 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
Radioligand Labeled Binding Assay and [35S]GTP-gamma-S Binding Assay from Article 10.1021/jm050921q: "Structure-activity relationships of bifunctional peptides based on overlapping pharmacophores at opioid and cholecystokinin receptors."
Assay data:19 Active, 6 Activity ≤ 1 nM, 18 Activity ≤ 1 µM, 19 Tested
PRESTO-Tango GPCRome screening (CCKBR)
CCKB (h) (CCK2) CEREP ligand profiling
CCK2 (human) CEREP ligand profiling
CCKB/H Cerep selectivity data (BI)
CCKB (CCK2) CEREP ligand profiling
CholecystokininB receptor (h) CEREP ligand profiling
CCKB (h) Ligand binding assay
CCKB (h) CEREP ligand profiling
hCCK2 Cerep panel
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