BioAssay by Target (List) for Gene (Select 9263) - PubChem BioAssay - NCBI

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Select item 19629641.

STK17A SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1962964

Summary Related BioAssays by Target

Select item 19628602.

STK17A SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1962860

Summary Related BioAssays by Target

Select item 19627623.

STK17A SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1962762

Summary Related BioAssays by Target

Select item 19626634.

STK17A SGC Tm panel (DSF)

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1962663

Summary Related BioAssays by Target

Select item 19609055.

Inhibition of DRAK1 (unknown origin) at 10 uM by biochemical hotspot kinase assay relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1960905

Summary PubMed Citation Related BioAssays by Target

Select item 19348356.

Inhibition of human partial length wild type DRAK1 expressed in bacterial system at 1 uM by KINOMEscan analysis relative to control

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1934835

Summary PubMed Citation Related BioAssays by Target

Select item 19139037.

Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000305b STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1913903

Summary Related BioAssays by Target

Select item 19139028.

Selectivity interaction (KinomeScan (DiscoverX)) EUB0000305b STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1913902

Summary Related BioAssays by Target

Select item 19139019.

Selectivity interaction (Enzymatic assay (Eurofins)) EUB0000305b STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913901

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191390010.

Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000305b STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913900

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191389911.

Selectivity interaction (Enzymatic assay) EUB0000305b STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913899

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191358412.

Selectivity interaction (Kinase panel (ProQinase)) EUB0000631a STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Tested

AID:: 1913584

Summary Related BioAssays by Target

Select item 191338613.

Selectivity interaction (Upstate Kinase Profiler service (Millipore)) EUB0000056c STK17A

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913386

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191259514.

Thermal Shift Assay. Domain: start/stop: V50-P350

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:27 Tested

AID:: 1912595

Summary Related BioAssays by Target

Select item 191101415.

Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as gibbs free energy change by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:2 Tested

AID:: 1911014

Summary PubMed Citation Related BioAssays by Target

Select item 191101316.

Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as change in entropy by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:2 Tested

AID:: 1911013

Summary PubMed Citation Related BioAssays by Target

Select item 191100517.

Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) transfected in HEK293T cells using NanoBRET NanoGlo as substrate incubated for 2 hrs by NanoBRET assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:5 Active, 5 Activity ≤ 1 µM, 7 Tested

AID:: 1911005

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191100218.

Inhibition of human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli using KKLNRTLSFAEPG peptide as substrate in presence of [gamma-33P]ATP by radiometric based scintillation proximity assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested

AID:: 1911002

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191100119.

Binding affinity to human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli by isothermal titration calorimetry

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested

AID:: 1911001

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 191099720.

Binding affinity to human N-terminal His-tagged/ TEV cleavage fused DRAK1 (39 to 369 residues) expressed in Escherichia coli assessed as change in melting temperature at 10 uM by SYPRO orange dye based DSF assay

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase 17A

Assay data:7 Tested

AID:: 1910997

Summary PubMed Citation Related BioAssays by Target

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Target

Proteins (4)
BioAssays with protein sequences specified as targets
RNAi Target, Active (8)
BioAssays with gene sequences specified as RNAi targets and the activity is active

BioActivity

Active Compounds (57)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (4)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (38)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (57)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations
Primary Screening (40)
Primary high-throughput BioAssays where the activity outcome is based on percentage inhibition from a single dose
Chemical Screens (204)
BioAssays reporting BioActivity of chemical reagents
RNAi Screens (44)
BioAssays reporting BioActivity of RNAi reagents

Assay Project (2)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (166)
BioAssays extracted from the literature
NIH MLP (3)
BioAssays deposited by the NIH Molecular Libraries Program
Other (78)
BioAssays deposited by other experimentalists

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BioAssay by Target (List) for Gene (Select 9263) (248)
PubChem BioAssay
Homo sapiens
Homo sapiens
Celera Genomics WGS human genome sequencing project

BioProject
BioProject Links for Protein (Select 119590842) (1)
BioProject
TAP2 transporter 2, ATP binding cassette subfamily B member [Homo sapiens]
TAP2 transporter 2, ATP binding cassette subfamily B member [Homo sapiens]
Gene ID:6891

Gene
Gene Links for GEO Profiles (Select 96333518) (1)
Gene

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