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Activation of GLP2 receptor transfected in human HEK293 cells assessed as increase in intracellular cAMP level at 1 nM
Assay data:1 Active, 2 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Binding affinity towards GLP-2 receptor in human HEK293 cells measured by fluorescence assay
Assay data:9 Active, 3 Activity ≤ 1 nM, 9 Activity ≤ 1 µM, 9 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
PRESTO-Tango GPCRome screening (GLP2R)
Assay data:1 Tested
SummaryRelated BioAssays by Target
Agonist activity at human GLP-2 receptor expressed in CHO-K1 cells assessed as cAMP induction by FRET assay
Assay data:2 Active, 2 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 2 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
RNAi screen for vemurafenib enhancer genes in BRAFV600 melanoma - Primary Screen
Assay data:790 Active, 18119 Tested
Summary
Agonist activity at human GLP2 receptor expressed in HEK293 cells assessed as increase in intracellular cAMP accumulation by AlphaScreen assay
Assay data:14 Active, 13 Activity ≤ 1 nM, 15 Activity ≤ 1 µM, 15 Tested
Antagonist activity at GLP2R (unknown origin) at 10 uM by cAMP accumulation based assay relative to control
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at GLP2R (unknown origin) at 10 uM by cAMP accumulation based assay relative to control
Human GLP-2 receptor (Glucagon receptor family)
Assay data:4 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Potency index, ratio of compound EC50 to compound 2 EC50 for human GLP2R expressed in HEK293 cells
Assay data:29 Tested
Agonist activity at human GLP2R expressed in HEK293 cells after 5 hrs by luciferase reporter gene assay
Assay data:93 Active, 79 Activity ≤ 1 nM, 95 Activity ≤ 1 µM, 95 Tested
Genome-wide siRNA screen of genes regulating the Lipopolysaccharide-induced TNF-alpha response in human macrophages_Primary screen TNF readout
Assay data:2853 Active, 18113 Tested
SummaryRelated BioAssays by Same Project
A screen to identify synthetic lethal interactions with E-cadherin in an MCF10A isogenic cell line
Assay data:2442 Active, 18052 Tested
SummaryPubMed Citation
A screen to identify genes that regulate lymphatic endothelial cell migration - Primary Screen
Assay data:1034 Active, 18120 Tested
SummaryRelated BioAssays by Depositor
Identification of proteins required for the processing of the EWS-FLI1 nascent transcript
Assay data:59220 Tested
InfectX: Pathogen infection siRNA screens
Assay data:115372 Tested
A whole genome RNAi screen highlights components of the ER/Golgi as a prominent source of resistance to immunotoxin-mediated cytotoxicity
Assay data:555 Active, 64752 Tested
RNAi screen for vorinostat resistance genes - Primary Screen
Assay data:450 Active, 18118 Tested
Druggable Genome siRNA Screen for Enhancers of Camptothecin in MDA-MB-231 Breast Cancer Cells
Assay data:167 Active, 26449 Tested
Positive ago-allosteric modulation of GLP2R overexpressed in human SE302 cells assessed as reduction of GLP2-induced cAMP level at 3 to 10 uM after 30 mins
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