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Agonist activity at rat TRPV1 heterologously expressed in CHO cells assessed as capsaicin-induced [45Ca2+] uptake by liquid scintillation counting
Assay data:20 Tested
SummaryPubMed CitationRelated BioAssays by Target
Partial antagonist activity at rat TRPV1 heterologously expressed in CHO cells assessed as inhibition of capsaicin-induced [45Ca2+] uptake by liquid scintillation counting
Assay data:2 Tested
Antagonist activity at rat TRPV1 heterologously expressed in CHO cells assessed as inhibition of capsaicin-induced [45Ca2+] uptake by liquid scintillation counting
Assay data:18 Active, 17 Activity ≤ 1 µM, 18 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Displacement of [3H]RTX from rat TRPV1 after 60 mins by competitive binding assay
Assay data:18 Active, 17 Activity ≤ 1 µM, 20 Tested
Displacement of [3H]RTX from human TRPV1 expressed in CHO cells after 60 mins by liquid scintillation counting analysis
Assay data:8 Active, 8 Activity ≤ 1 µM, 8 Tested
Agonist activity at human TRPV1 expressed in CHO cells assessed as 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
Assay data:4 Active, 2 Activity ≤ 1 nM, 4 Activity ≤ 1 µM, 8 Tested
Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of RTX-induced 45Ca2+ uptake after 20 mins by liquid scintillation counting analysis
Assay data:4 Active, 4 Activity ≤ 1 µM, 8 Tested
Agonist activity at TRPV1 (unknown origin) relative to capsaicin
Assay data:1 Tested
Displacement of [3H]RTX from rat TRPV1 expressed in CHO cells
Assay data:10 Active, 1 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptake
Assay data:4 Active, 4 Activity ≤ 1 µM, 10 Tested
Agonist activity at rat TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptake relative to capsaicin
Assay data:3 Tested
Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-stimulated Ca2+ uptake
Assay data:6 Active, 6 Activity ≤ 1 µM, 10 Tested
Antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-stimulated Ca2+ uptake relative to control
Displacement of [3H]RTX from human TRPV1 expressed in CHO cells
Assay data:12 Active, 12 Activity ≤ 1 µM, 12 Tested
Agonist activity at human TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptake
Assay data:6 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 12 Tested
Agonist activity at human TRPV1 expressed in CHO cells assessed as stimulation of Ca2+ uptake relative to capsaicin
Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-stimulated Ca2+ uptake
Assay data:7 Active, 5 Activity ≤ 1 µM, 11 Tested
Antagonist activity at human TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-stimulated Ca2+ uptake relative to control
Partial antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-stimulated Ca2+ uptake
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Partial antagonist activity at rat TRPV1 expressed in CHO cells assessed as inhibition of capsaicin-stimulated Ca2+ uptake measured as residual agonism
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