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Antagonist activity at recombinant human GABA-A rho-1 receptor transiently expressed in human tsA201 cells incubated for 30 mins and measured up to 90 secs by FMP dye based FLIPR membrane potential blue assay
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Agonist activity at recombinant human GABA-A rho-1 receptor transiently expressed in human tsA201 cells at 300 uM incubated for 30 mins and measured up to 90 secs by FMP dye based FLIPR membrane potential blue assay
Agonist activity at recombinant human GABA-A rho-1 receptor transiently expressed in human tsA201 cells at >= 100 uM incubated for 30 mins and measured up to 90 secs by FMP dye based FLIPR membrane potential blue assay
Assay data:4 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Agonist activity at recombinant human GABA-A rho-1 receptor transiently expressed in human tsA201 cells assessed as GABA-induced maximum response incubated for 30 mins and measured up to 90 secs by FMP dye based FLIPR membrane potential blue assay relative to GABA
Assay data:12 Tested
Agonist activity at recombinant human GABA-A rho-1 receptor transiently expressed in human tsA201 cells incubated for 30 mins and measured up to 90 secs by FMP dye based FLIPR membrane potential blue assay
Assay data:10 Active, 1 Activity ≤ 1 µM, 13 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Rat GABAA receptor rho1 subunit (GABAA receptors)
Assay data:1 Active, 1 Tested
Human GABAA receptor rho2 subunit (GABAA receptors)
Assay data:13 Active, 13 Tested
Human GABAA receptor rho1 subunit (GABAA receptors)
Human GABAA receptor rho3 subunit (GABAA receptors)
Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assay relative to GABA
Assay data:5 Tested
Agonist activity at human GABAA rho1 expressed in tsA-201cells at 1 mM by FLIPR membrane potential blue assay
Assay data:2 Active, 2 Tested
Agonist activity at human GABAA rho1 expressed in tsA-201cells by FLIPR membrane potential blue assay
Assay data:8 Active, 2 Activity ≤ 1 µM, 20 Tested
Displacement of [3H]EBOB from recombinant Homo sapiens (human) GABA rho1 receptor
Assay data:2 Active, 2 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Inhibition of human GABA C receptor subunit rho-1 receptor expressed in Xenopus laevis oocytes assessed as inhibition of GABA-induced current at 3 uM by two-electrode voltage clamp method
Assay data:2 Tested
Antagonist activity at human recombinant GABAA rho1 receptor expressed in Xenopus laevis assessed as inhibition of GABA-induced chloride current production at 300 uM after 2 to 5 days by two-electrode voltage-clamp electrophysiological assay relative to control
Antagonist activity at human recombinant GABAA rho1 receptor expressed in Xenopus laevis assessed as inhibition of GABA-induced chloride current production after 2 to 5 days by two-electrode voltage-clamp electrophysiological assay
Assay data:2 Active, 8 Tested
Activity at human recombinant GABA(C) receptor expressed in Xenopus oocytes assessed as effect on GABA-induced activation at 3 uM by two-electrode voltage clamp technique relative to control
Assay data:1 Tested
Agonist activity at GABAC rho1 receptor (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 3 Tested
Partial agonist activity at GABAC rho1 receptor (unknown origin)
Antagonist activity at GABAC rho1 receptor (unknown origin)
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