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Enzyme Assay from US Patent US11884671: "Purinone compounds and their use in treating cancer"
Assay data:51 Tested
SummaryRelated BioAssays by DepositorRelated BioAssays by Target
Assay data:1 Active, 51 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
TTK Enzyme Assay from US Patent US11884671: "Purinone compounds and their use in treating cancer"
Assay data:46 Active, 22 Activity ≤ 1 µM, 51 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
HPK1 Kinase Assay (Biochemical Assay) from US Patent US20240025922: "TETRAHYDROPYRIDO[3,4-d]PYRIMIDINES AS HPK1 INHIBITORS"
Assay data:181 Active, 187 Activity ≤ 1 µM, 187 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
RIPK1-ADP-Glo Enzymatic Assay from US Patent US20240025912: "RIPK1 INHIBITORS AND METHODS OF USE"
Assay data:108 Active, 108 Activity ≤ 1 µM, 108 Tested
Inhibitory Activity of the Compounds of the Invention Against ROS1, NTRK and ALK and their Drug-Resistant Kinases from US Patent US20240025908: "COMPOUND USED AS KINASE INHIBITOR AND USE THEREOF"
Assay data:29 Active, 14 Activity ≤ 1 nM, 29 Activity ≤ 1 µM, 29 Tested
In Vitro SIK2 Kinase Assay from US Patent US20240025892: "SALT INDUCIBLE KINASE INHIBITORS"
Assay data:66 Active, 5 Activity ≤ 1 nM, 63 Activity ≤ 1 µM, 66 Tested
Biochemical Assay from US Patent US20240025884: "COMPOUNDS AS GCN2 INHIBITORS, PHARMACEUTICAL COMPOSITIONS AND USES THEREOF"
Assay data:498 Active, 503 Activity ≤ 1 µM, 503 Tested
HTRF Assay from US Patent US20240018153: "BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF"
Assay data:13 Active, 13 Activity ≤ 1 µM, 13 Tested
Assay data:10 Active, 10 Activity ≤ 1 µM, 10 Tested
Assay data:11 Active, 11 Activity ≤ 1 µM, 11 Tested
Assay data:9 Active, 9 Activity ≤ 1 µM, 9 Tested
In Vitro Kinase Detection Assay from US Patent US20240018147: "SALT OF COMPOUND FOR DEGRADING BTK, CRYSTAL FORM THEREOF, AND USE THEREOF IN MEDICINE"
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
In vitro Assay from US Patent US20240018122: "PYRIDAZINYL AMINO DERIVATIVES AS ALK5 INHIBITORS"
Assay data:187 Active, 157 Activity ≤ 1 nM, 186 Activity ≤ 1 µM, 188 Tested
Reaction Biology 33P Hotspot assay from US Patent US20240010634: "PYRIMIDINYL SULFONAMIDES AS INHIBITORS OF ACK1/TNK2 TYROSINE KINASE"
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Biochemical Assay for Inhibitors of CLK2 Kinase Activity Assay from US Patent US11866436: "Benzo[c][2,6]naphthyridine derivatives, compositions and therapeutic uses thereof"
Assay data:181 Active, 131 Activity ≤ 1 µM, 181 Tested
Biochemical Assay for Inhibitors of CK2α Kinase Activity Assay from US Patent US11866436: "Benzo[c][2,6]naphthyridine derivatives, compositions and therapeutic uses thereof"
Assay data:181 Active, 118 Activity ≤ 1 nM, 181 Activity ≤ 1 µM, 181 Tested
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