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Displacement of [3H]Me-TRH from human recombinant TRH receptor at 10 uM after 120 mins by scintillation counting analysis relative to control
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Thyrotropin Releasing Hormone (TRH) Eurofins-Panlabs radioligand binding assay
Assay data:4 Tested
SummaryRelated BioAssays by Target
Inhibition of rat TRH receptor at 10 uM relative to control
Activity at human TRH receptor up to 10 uM
Assay data:2 Tested
Thyrotropin-releasing hormone receptor (TRHR) small molecule antagonists: Summary
Assay data:130 Active, 9667 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Thyrotropin-releasing hormone receptor (TRHR) small molecule agonists: Summary
Assay data:94 Active, 9667 Tested
qHTS assay to identify small molecule agonists of the thyrotropin-releasing hormone receptor (TRHR) signaling pathway
Assay data:85 Active, 5 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule antagonists of the thyrotropin-releasing hormone receptor (TRHR) signaling pathway
Assay data:81 Active, 11 Activity ≤ 1 µM, 9667 Tested
Human TRH1 receptor (Thyrotropin-releasing hormone receptors)
Assay data:2 Active, 2 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Mouse TRH1 receptor (Thyrotropin-releasing hormone receptors)
Assay data:1 Active, 1 Tested
Rat TRH1 receptor (Thyrotropin-releasing hormone receptors)
Assay data:4 Active, 4 Tested
Displacement of [3H]-3MeHis-TRH from TRH receptor in Sprague-Dawley rat cortical membranes
Assay data:2 Active, 1 Activity ≤ 1 µM, 3 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Displacement of [3H]-Me-His-TRH from mouse TRH-R1 expressed in HEK293 cell membranes at 30 uM after 4 hrs by scintillation counting method
Displacement of [2,5-125I2]-Me-His-TRH from wild type TRHR mouse brain membranes at 0.3 uM after 4 hrs by scintillation counting method
Displacement of [2,5-125I2]-Me-His-TRH from wild type TRHR mouse brain membranes at 1 uM after 4 hrs by scintillation counting method
Displacement of [2,5-125I2]-Me-His-TRH from wild type TRHR mouse brain membranes at 3 uM after 4 hrs by scintillation counting method
Displacement of [2,5-125I2]-Me-His-TRH from wild type TRHR mouse brain membranes at 10 uM after 4 hrs by scintillation counting method
Displacement of [2,5-125I2]-Me-His-TRH from wild type TRHR mouse brain membranes at 30 uM after 4 hrs by scintillation counting method
Displacement of [3H]-Me-His-TRH from wild type TRHR mouse brain membrane at 3 uM after 4 hrs by scintillation counting method
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