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Adrenomedullin AM1 Eurofins-Panlabs radioligand binding assay
Assay data:2 Tested
SummaryRelated BioAssays by Target
Calcitonin Eurofins-Panlabs radioligand binding assay
Assay data:3 Tested
PRESTO-Tango GPCRome screening (CALCRb)
Assay data:1 Tested
Antagonist activity at human adrenomedullin-1 receptor
SummaryPubMed CitationRelated BioAssays by Target
Antagonist activity at human amylin-1 receptor
Agonist activity at eYFP-tagged CLR/eCFP-tagged RAMP2-derived AM1 receptor (unknown origin) expressed in HEK293 cells assessed as cAMP accumulation after 3 hrs by ONE-Glo substrate-based luminescence assay
Assay data:4 Tested
Displacement of [125I]-labeled human calcitonin from human calcitonin receptor expressed in BHK tkts13 whole cells incubated for 60 mins by scintillation proximity assay
Assay data:91 Active, 50 Activity ≤ 1 nM, 91 Activity ≤ 1 µM, 91 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Displacement of [125I]-labeled rat amylin from human amylin receptor expressed in BHK tkts13 whole cells co-expressing RAMP3 incubated for 60 mins by scintillation proximity assay
Assay data:91 Active, 48 Activity ≤ 1 nM, 91 Activity ≤ 1 µM, 91 Tested
Displacement of [125I]-labeled rat calcitonin from human calcitonin receptor expressed in BHK tkts13 cell membranes incubated for 1 hr by scintillation proximity assay
Assay data:35 Active, 35 Activity ≤ 1 nM, 35 Activity ≤ 1 µM, 39 Tested
Displacement of [125I]-labeled rat amylin from rat amylin receptor expressed in BHK tkts13 cell membranes co-expressing RAMP3 incubated for 120 mins by scintillation proximity assay
Assay data:33 Active, 29 Activity ≤ 1 nM, 33 Activity ≤ 1 µM, 39 Tested
Displacement of [125I]-labeled human calcitonin from human calcitonin receptor expressed in BHK tkts13 cell membranes incubated for 1 hr by scintillation proximity assay
Assay data:39 Active, 39 Activity ≤ 1 nM, 39 Activity ≤ 1 µM, 39 Tested
Displacement of [125I]-labeled rat amylin from human amylin receptor expressed in BHK570 cell membranes co-expressing RAMP3 incubated for 120 mins by scintillation proximity assay
Agonist activity at human calcitonin receptor expressed in BHK570 cells assessed as increase in intracellular cAMP concentration incubated for 3 hrs in presence of 10% FBS by CRE luciferase reporter gene assay
Assay data:96 Active, 96 Activity ≤ 1 nM, 96 Activity ≤ 1 µM, 96 Tested
Agonist activity at human amylin receptor expressed in BHK570 cells co-expressing RAMP3 assessed as increase in intracellular cAMP concentration incubated for 3 hrs in presence of 10% FBS by CRE luciferase reporter gene assay
Agonist activity at human calcitonin receptor expressed in BHK570 cells assessed as increase in intracellular cAMP concentration incubated for 3 hrs in absence of albumin by CRE luciferase reporter gene assay
Assay data:141 Active, 141 Activity ≤ 1 nM, 141 Activity ≤ 1 µM, 143 Tested
Agonist activity at human amylin receptor expressed in BHK570 cells co-expressing RAMP3 assessed as increase in intracellular cAMP concentration incubated for 3 hrs in absence of albumin by CRE luciferase reporter gene assay
Assay data:141 Active, 140 Activity ≤ 1 nM, 141 Activity ≤ 1 µM, 143 Tested
Human CT receptor (Calcitonin receptors)
Assay data:11 Active, 11 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of human calcitonin receptor at 10 uM relative to control
Displacement of [125I]calcitonin from human CT receptor expressed in HEK293 cells
Assay data:1 Active, 1 Tested
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