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Selectivity interaction (KinomeScan (DiscoverX)) EUB0000704a WNK3
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of WNK3 (unknown origin) at 10 uM relative to control
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of WNK3 (unknown origin) at 1 uM
WNK3 DiscoveRx kinase panel
WNK3(h) Kinase panel
Inhibition of human recombinant WNK3 assessed as reduction in substrate phosphorylation at 500 nM using ATP and Ulight-CKKSRGDYMTMQIG (IRS-1) incubated for 60 min by LANCE detection method
WNK In Vitro Radiometric Assays from Article 10.1021/acschembio.6b00511: "Discovery and Characterization of Allosteric WNK Kinase Inhibitors."
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
KinomeScan assay: inhibition of WNK3
Assay data:1 Active, 108 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
WNK3(h) Eurofins kinase panel
WNK3 ProQinase selectivity panel
WNK3(h) Eurofins Kinase panel
WNK3 (h) Millipore kinase activity assay
WNK3(h) Millipore kinase panel
WNK lysine deficient protein kinase 3 Millipore kinase panel
WNK3 Invitrogen Lab (UK) kinase screen (BI)
Inhibition of WNK3 (unknown origin) assessed as residual activity measured at 1 uM
Assay data:3 Tested
Inhibition of human WNK3 assessed as percent of control at 2000 nM by KINOMEscan assay relative to control
Inhibition of human WNK3 assessed as percent of control at 1000 nM by KINOMEscan assay relative to control
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