Related BioAssays, by Target Similarity (List) for PubChem BioAssay (S - PubChem BioAssay - NCBI

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Select item 19125131.

Thermal Shift Assay. Domain: start/stop: M1-S424

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:27 Tested

AID:: 1912513

Summary Related BioAssays by Target

Select item 18356472.

MRCKB DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:1 Tested

AID:: 1835647

Summary Related BioAssays by Target

Select item 18354683.

MRCKA DiscoveRx kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Tested

AID:: 1835468

Summary Related BioAssays by Target

Select item 18350554.

MRCKbeta(h) Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:1 Tested

AID:: 1835055

Summary Related BioAssays by Target

Select item 18350545.

MRCKalpha(h) Kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Tested

AID:: 1835054

Summary Related BioAssays by Target

Select item 18342276.

Inhibition of MRCKbeta (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:1 Tested

AID:: 1834227

Summary PubMed Citation Related BioAssays by Target

Select item 18342267.

Inhibition of MRCKalpha (unknown origin) at 1 uM

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Tested

AID:: 1834226

Summary PubMed Citation Related BioAssays by Target

Select item 18068318.

Kinase Assay from US Patent US11447505: "Pyrrolo[2,3-b]pyridine compounds and their use in the treatment of cancer"

Source:: BindingDB

Protein Targets:: Rho-associated protein kinase 1; ...
Total:: 4

Assay data:225 Active, 76 Activity ≤ 1 nM, 225 Activity ≤ 1 µM, 225 Tested

AID:: 1806831

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 17998049.

Binding Assay from Article 10.1074/jbc.M707463200: "Characterization of the interaction of phorbol esters with the C1 domain of MRCK (myotonic dystrophy kinase-related Cdc42 binding kinase) alpha/beta."

Source:: BindingDB

Protein Targets:: Protein kinase C alpha type; ...
Total:: 4

Assay data:5 Active, 2 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested

AID:: 1799804

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 179856010.

MRCK Inhibition Assay from Article 10.1021/jm800986w: "Discovery of substituted 4-(pyrazol-4-yl)-phenylbenzodioxane-2-carboxamides as potent and highly selective Rho kinase (ROCK-II) inhibitors."

Source:: BindingDB

Protein Targets:: Serine/threonine-protein kinase MRCK alpha; ...
Total:: 1

Assay data:5 Active, 1 Activity ≤ 1 µM, 5 Tested

AID:: 1798560

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Depositor Related BioAssays by Target

Select item 179420611.

KinomeScan assay: inhibition of MRCKB

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:108 Tested

AID:: 1794206

Summary Related BioAssays by Target

Select item 179420512.

KinomeScan assay: inhibition of MRCKA

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:108 Tested

AID:: 1794205

Summary Related BioAssays by Target

Select item 179360613.

MRCKalpha(CD4ALGY1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793606

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179331514.

MRCKalpha(CD4ALGY1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793315

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179302115.

MRCKalpha(CD4ALGY1) Takeda global kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Activity ≤ 1 µM, 1 Tested

AID:: 1793021

Summary Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 179275916.

MRCKbeta(h) Eurofins kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:1 Tested

AID:: 1792759

Summary Related BioAssays by Target

Select item 179275817.

MRCKalpha(h) Eurofins kinase panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Tested

AID:: 1792758

Summary Related BioAssays by Target

Select item 179221418.

CDC42BPB ProQinase selectivity panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:1 Tested

AID:: 1792214

Summary Related BioAssays by Target

Select item 179221319.

CDC42BPA ProQinase selectivity panel

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK alpha

Assay data:1 Tested

AID:: 1792213

Summary Related BioAssays by Target

Select item 179094720.

CDC42 BPB (MRCKB) Kinase screen

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase MRCK beta

Assay data:1 Tested

AID:: 1790947

Summary Related BioAssays by Target

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Target

Proteins (4)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (32)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (5)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (28)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Confirmatory (41)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Literature Extraction (193)
BioAssays extracted from the literature
NIH MLP (1)
BioAssays deposited by the NIH Molecular Libraries Program
Other (46)
BioAssays deposited by other experimentalists

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Related BioAssays, by Target Similarity (List) for PubChem BioAss... (240)
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PubChem BioAssay
Profile neighbors for GEO Profiles (Select 132351089) (174)
GEO Profiles
Chromosome neighbors for GEO Profiles (Select 132349781) (20)
GEO Profiles
Chromosome neighbors for GEO Profiles (Select 129873854) (20)
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CCT8 chaperonin containing TCP1 subunit 8 [Homo sapiens]
CCT8 chaperonin containing TCP1 subunit 8 [Homo sapiens]
Gene ID:10694

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