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8-[Fluo]-cAMP Fluorescence Polarization Binding Assay from Article 10.1021/acs.biochem.6b01152: "Electrostatic Interactions as Mediators in the Allosteric Activation of Protein Kinase A RIa."
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Activation of recombinant human PKAR1alpha expressed in Escherichia coli using Kemptide as substrate by spectrophotometric method
Assay data:5 Active, 5 Activity ≤ 1 µM, 5 Tested
Binding affinity to recombinant human full length PKA-R1beta expressed in Escherichia coli BL21 DE3-RIL cells assessed as reduction in interaction with AKAP at 20 nM by fluorescence polarization analysis
Assay data:13 Tested
SummaryPubMed CitationRelated BioAssays by Target
Binding affinity to recombinant human full length PKA-R1alpha expressed in Escherichia coli BL21 DE3-RIL cells assessed as reduction in interaction with AKAP at 20 nM by fluorescence polarization analysis
Late-stage fluorescence polarization-based biochemical dose response assay for activators of the Protein Kinase A-R1A (PKA-R1A) complex.
Assay data:9 Tested
SummaryPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Counterscreen for activators of the Protein Kinase A-R2B (PKA-R2B) complex: fluorescence polarization-based biochemical high throughput dose response assay to identify activators of the Protein Kinase A-R1A (PKA-R1A) complex
Assay data:7 Active, 3 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Fluorescence polarization-based biochemical high throughput dose response assay for activators of the Protein Kinase A-R1A (PKA-R1A) complex
Assay data:7 Active, 3 Activity ≤ 1 µM, 8 Tested
Fluorescence polarization-based biochemical high throughput confirmation assay for activators of the Protein Kinase A-R1A (PKA-R1A) complex
Assay data:27 Active, 276 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
Counterscreen for activators of the Protein Kinase A-R1A (PKA-R1A) complex: fluorescence polarization-based biochemical high throughput screening assay to identify fluorescence polarization assay artifacts
Assay data:19 Active, 276 Tested
Fluorescence polarization-based biochemical primary high throughput screening assay to identify activators of the Protein Kinase A-R1A (PKA-R1A) complex
Assay data:285 Active, 343700 Tested
Summary of the probe development efforts to identify activators of the Protein Kinase A-R1A (PKA-R1A) complex
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