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Assay of Inhibition of Escherichia coli RNA Polymerase from US Patent US10800725: "Arylpropionyl-triketone antibacterial agents"
Assay data:16 Active, 7 Activity ≤ 1 µM, 20 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Stimulation of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP by scintillation counting
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP by scintillation counting
Assay data:1 Tested
Stimulation of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 25 ug/ml by scintillation counting
Inhibition of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 25 ug/ml by scintillation counting
Assay data:4 Tested
Stimulation of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 50 ug/ml by scintillation counting
Inhibition of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 50 ug/ml by scintillation counting
Stimulation of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 100 ug/ml by scintillation counting
Inhibition of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 100 ug/ml by scintillation counting
Stimulation of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 200 ug/ml by scintillation counting
Inhibition of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 200 ug/ml by scintillation counting
Stimulation of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 400 ug/ml by scintillation counting
Inhibition of Escherichia coli DNA-primed RNA polymerase activity using [8-14C]ATP at 400 ug/ml by scintillation counting
Inhibition of Escherichia coli DNA-dependent RNA polymerase assessed as [3H]UMP incorporation into RNA using calf thymus DNA at 0.12 mM by liquid scintillation counting
Assay data:3 Active, 3 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of Escherichia coli DNA-dependent RNA polymerase
Inhibition of Escherichia coli DNA-dependent RNA polymerase at 0.05 ug/ml using Micrococcus luteus DNA as primer
Inhibition of Escherichia coli DNA-dependent RNA polymerase at 0.05 ug/ml using calf thymus DNA as primer
Inhibition of Escherichia coli DNA-dependent RNA polymerase at 0.1 ug/ml using Micrococcus luteus DNA as primer
Inhibition of Escherichia coli DNA-dependent RNA polymerase at 0.1 ug/ml using calf thymus DNA as primer
Inhibition of Escherichia coli DNA-dependent RNA polymerase at 0.25 ug/ml using Micrococcus luteus DNA as primer
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