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In vitro PDE4B Enzyme Activity Detection Assay from US Patent US20240083921: "BORATE DERIVATIVE AND USES THEREOF"
Assay data:14 Active, 12 Activity ≤ 1 nM, 14 Activity ≤ 1 µM, 14 Tested
SummaryRelated BioAssays by Target
PDE3B Enzyme Inhibition from US Patent US11897867: "6-phenyl-4,5-dihydropyridazin-3(2H)-one derivatives as PDE3A and PDE3B inhibitors for treating cancer"
Assay data:129 Active, 130 Activity ≤ 1 µM, 130 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Cross screening panel
Assay data:1 Tested
Safety47 Scan (DiscoverX - Eurofins)
Phosphodiesterase PDE5 Eurofins Panlabs panel
Phosphodiesterase PDE4 Eurofins Panlabs panel
Phosphodiesterase PDE3 Eurofins Panlabs panel
Panlabs assay PDE10A2
Panlabs assay PDE9A2
Panlabs assay PDE8A1
Panlabs assay PDE7B
Panlabs assay PDE7A
Panlabs assay PDE6
Panlabs assay PDE5A
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