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Selectivity interaction (KinomeScan (DiscoverX)) EUB0000750a CIT
Assay data:1 Tested
SummaryRelated BioAssays by Target
Inhibition of human CIT at 100 nM by KINOMEscan assay relative to control
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of CRIK (unknown origin)
Assay data:5 Active, 3 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of human CRIK at 1 uM relative to control
Inhibition of wild-type human partial length CIT (M68 to E432 residues) expressed in bacterial expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control
CIT DiscoveRx kinase panel
CRIK(h) Kinase panel
Inhibition of STK21 (unknown origin) at 1 uM
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
KinomeScan assay: inhibition of CIT
Assay data:1 Active, 108 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
CRIK(CIT1LGY1) Takeda global kinase panel
Assay data:1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by Target
CRIK(h) Millipore kinase panel
Inhibition of human STK21 using MBP as substrate assessed as enzyme activity incubated for 2 hrs by [gamma-33P]-ATP assay relative to control
Inhibition of CRIK (unknown origin) by Kinomescan method
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Inhibition of CRIK (unknown origin) assessed as residual binding level at 1 uM by Kinomescan method relative to control
Inhibition of human CIT assessed as percent of control at 2000 nM by KINOMEscan assay relative to control
Inhibition of DNA-tagged human CIT assessed as percent of control at 50000 nM by qPCR analysis relative to control
Inhibition of human CIT assessed as percent of control at 1000 nM by KINOMEscan assay relative to control
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