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Inhibition of PACE4 (unknown origin)
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of recombinant soluble human PACE4 using pyroGlu-Arg-Thr-Lys-Arg-methyl-coumaryl-7-amide as substrate measured after 1 hr
Assay data:4 Active, 4 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of recombinant C-terminal truncated human SPC4 expressed in drosophila Schneider 2 cells after 1 hr by spectrofluorometry
Inhibition of recombinant human PACE4 expressed in drosophila S2 cells using pyrGlu-Arg-Thr-Lys-Arg-7-amido-4-methylcoumarin as substrate after 60 mins by spectrofluorometry method
Assay data:75 Active, 9 Activity ≤ 1 nM, 75 Activity ≤ 1 µM, 75 Tested
Inhibition of recombinant human PACE4 using pGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate by spectrofluorometry
Assay data:12 Active, 12 Activity ≤ 1 µM, 12 Tested
Inhibition of recombinant human PACE4 expressed in S2 insect cells using pyroGlu-Arg-Thr-Lys-Arg-AMC peptide as substrate after 1 hr by spectrofluorometry
Assay data:27 Active, 27 Activity ≤ 1 µM, 27 Tested
Inhibition of human recombinant PACE4 expressed in drosophila schneider 2 cells using pyroGlu-Arg-Thr-Lys-Arg-AMC as substrate after 1 hr
Assay data:19 Active, 18 Activity ≤ 1 µM, 21 Tested
Competitive inhibition of human recombinant PACE4 expressed in Drosophila S2 cells using pyroGlu-Arg-Val-Lys-Arg-methyl-coumaryl-7-amide as substrate at pH 6.5 after 60 mins by spectrofluorometric analysis
Assay data:16 Active, 2 Activity ≤ 1 nM, 14 Activity ≤ 1 µM, 17 Tested
Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assay
Assay data:5 Active, 1 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested
Inhibition of rat PACE4 up to 100 uM
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of rat PACE4 assessed as fluorescent Pyr-RTKR-AMC substrate cleavage
Assay data:6 Active, 5 Activity ≤ 1 µM, 6 Tested
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