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Inhibition of wild type human YSK4 in presence of ATP by radiometric kinase assay
Assay data:1 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of wild type human YSK4 at 1 uM by DiscoverX scanMAX assay relative to control
Inhibition of YSK4 (unknown origin) assessed as dissociation constant
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of YSK4 (unknown origin) at 1 uM relative to control
Assay data:3 Tested
In Vitro Effect Assay from US Patent US11608319: "Beta-amino acid derivative, kinase inhibitor and pharmaceutical composition containing the same, and method for performing an in vivo related application that benefits from the inhibition of a kinase"
Assay data:7 Activity ≤ 1 µM, 15 Tested
SummaryCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
Selectivity interaction (Kinase Panel (competition binding assay)) EUB0000589aTFA MAP3K19
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000138c MAP3K19
SummaryRelated BioAssays by Target
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000702a MAP3K19
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000701a MAP3K19
Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000305b MAP3K19
Selectivity interaction (KinomeScan (DiscoverX)) EUB0000305b MAP3K19
Selectivity interaction (KinomeScan (DiscoverX, competition-binding assay)) EUB0000305b MAP3K19
Inhibition of wild-type human partial length YSK4 (T1019 to H1328 residues) expressed in mammalian expression system at 10 uM by Kinomescan method relative to control
Inhibition of wild-type human partial length YSK4 (T1019 to H1328 residues) expressed in mammalian expression system assessed as residual binding level at 1 uM by Kinomescan method relative to control
YSK4 DiscoveRx kinase panel
Inhibition of YSK4 (unknown origin) at 1 uM
Inhibition of YSK4 (unknown origin) at 1 uM by kinome scan method
Assay data:1 Active, 1 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Inhibition of wild-type human partial length YSK4 (T1019 to H1328 residues) expressed in mammalian expression system at 1 uM by Kinomescan method
KinomeScan assay: inhibition of YSK4
Assay data:4 Active, 108 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
NanoBRET with MAP3K19
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