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Antagonist activity at human TBXA2R in an in vitro cell-based assay measured by fluorescence spectroscopy
Assay data:8 Active, 1 Activity ≤ 1 µM, 71 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Binding affinity towards human TBXA2R in an in vitro assay with cellular components measured by scintillation proximity assay
Assay data:14 Active, 2 Activity ≤ 1 µM, 1022 Tested
Assay data:34 Active, 15 Activity ≤ 1 µM, 906 Tested
Agonist activity at human TBXA2R in an in vitro cell-based assay (CRO assay) measured by fluorescence spectroscopy
Assay data:13 Active, 8 Activity ≤ 1 µM, 927 Tested
Agonist activity at human TBXA2R in an in vitro cell free assay (NIBR assay) measured by fluorescent imaging plate reader
Assay data:71 Tested
SummaryPubMed CitationRelated BioAssays by Target
Selectivity interaction (Prostanoid receptor binding assay) EUB0000334a TBXA2R
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Selectivity interaction (Prostanoid receptor binding assay) EUB0000297b TBXA2R
Cell Based Assay from US Patent US9422273: "Compounds act at multiple prostaglandin receptors giving a general anti-inflammatory response"
Assay data:5 Active, 5 Activity ≤ 1 nM, 5 Activity ≤ 1 µM, 5 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
FLIPR Assay from US Patent US9394273: "Therapeutic prostaglandin receptor agonists"
Assay data:10 Active, 4 Activity ≤ 1 µM, 10 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Target
PRESTO-Tango GPCRome screening (TBXA2R)
Assay data:1 Tested
SummaryRelated BioAssays by Target
TXA2/P GH2 (h)(TP) CEREP ligand profiling
Binding assay (TBXA2R)
Prostanoid receptor binding assay (TBXA2R)
Assay data:2 Tested
PROST_A2TP Eurofins-Panlabs selectivity data (BI)
TXA2/PGH2 CEREP ligand profiling
Thromboxane A2/ prostaglandin H2 receptors CEREP ligand profiling
TXA2/PGH2 (h) Ligand binding assay
Eurofins-Panlabs cell assay (ID:338490)
Inhibition of human thromboxane A2 at 0.1 to 1 uM
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