Related BioAssays, by Target Similarity (List) for PubChem BioAssay (S - PubChem BioAssay - NCBI

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Select item 19583081.

Binding affinity to human partial length PCAF (G715 to D831 residues) expressed in bacterial expression system by BROMOscan assay

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:4 Tested

AID:: 1958308

Summary PubMed Citation Related BioAssays by Target

Select item 19583052.

Binding affinity to human partial length GCN5L2 (E726 to K837 residues) expressed in bacterial expression system by BROMOscan assay

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:2 Active, 2 Activity ≤ 1 µM, 4 Tested

AID:: 1958305

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19491543.

Displacement of biotinylated JQ1 from PCAF bromodomain (unknown origin) incubated for 20 mins by AlphaLISA assay

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Tested

AID:: 1949154

Summary PubMed Citation Related BioAssays by Target

Select item 19491464.

Binding affinity to PCAF bromodomain (unknown origin) incubated for 60 mins by TR-FRET assay

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Tested

AID:: 1949146

Summary PubMed Citation Related BioAssays by Target

Select item 19427575.

PROTAC activity at PCAF/CRBN in human THP-1 cells

Source:: ChEMBL

Protein Targets:: Histone acetyltransferase KAT2B; ...
Total:: 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1942757

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19331316.

Binding affinity to PCAF (unknown origin) assessed as change in melting temperature at 200 uM incubated for 30 to 60 mins by SYPRO orange dye based thermal shift assay

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:2 Tested

AID:: 1933131

Summary PubMed Citation Related BioAssays by Target

Select item 19292547.

Inhibition of GST-tagged PCAF bromodomain (719 to 832 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) using Biotin-GISYGR-AcK-KKRRQRRRP as substrate incubated for 12 hrs by ELISA

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Active, 1 Tested

AID:: 1929254

Summary Compounds, Active PubMed Citation Related BioAssays by Target

Select item 19185038.

Inhibition of pCAF (unknown origin) using Histone H3 substrate at 1 uM relative to control

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Tested

AID:: 1918503

Summary PubMed Citation Related BioAssays by Target

Select item 19185009.

Inhibition of GCN5 (unknown origin) using Histone H3 substrate at 1 uM relative to control

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:1 Tested

AID:: 1918500

Summary PubMed Citation Related BioAssays by Target

Select item 191486410.

Selectivity interaction (TR-FRET assay) EUB0000256b KAT2B

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Tested

AID:: 1914864

Summary Related BioAssays by Target

Select item 191485211.

Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000253b KAT2B

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Tested

AID:: 1914852

Summary Related BioAssays by Target

Select item 191485112.

Selectivity interaction (BROMOscan? panel (DiscoverX)) EUB0000253b KAT2B

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914851

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191485013.

Selectivity interaction (Bromodomain panel (DSF assay)) EUB0000253b KAT2B

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Tested

AID:: 1914850

Summary Related BioAssays by Target

Select item 191484914.

Selectivity interaction (NanoBRET assay (HEK293T cells)) EUB0000253b KAT2A

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:1 Tested

AID:: 1914849

Summary Related BioAssays by Target

Select item 191484815.

Selectivity interaction (BROMOscan? panel (DiscoverX)) EUB0000253b KAT2A

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1914848

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191470816.

Selectivity interaction (HAT panel) EUB0000329a KAT2A

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:1 Tested

AID:: 1914708

Summary Related BioAssays by Target

Select item 191329717.

Affinity Biochemical interaction (Bromoscan assay (DiscoverX)) EUB0000256b KAT2B

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913297

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191329618.

Affinity Biochemical interaction (Bromoscan assay (DiscoverX)) EUB0000256b KAT2A

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913296

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191326819.

Affinity Biochemical interaction (BROMOscan assay (DiscoverX)) EUB0000218c KAT2B

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2B

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913268

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

Select item 191326720.

Affinity Biochemical interaction (BROMOscan assay (DiscoverX)) EUB0000218c KAT2A

Source:: ChEMBL

Protein Target:: Histone acetyltransferase KAT2A

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1913267

Summary Compounds, Active Compounds, activity ≤ 1 µM Related BioAssays by Target

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Proteins (4)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (90)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (2)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (45)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (150)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Assay Project (3)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

Depositor Category

Literature Extraction (253)
BioAssays extracted from the literature
NIH MLP (3)
BioAssays deposited by the NIH Molecular Libraries Program
Other (33)
BioAssays deposited by other experimentalists

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