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Selectivity interaction (CEREP panel (Eurofins, panel of ion channels, receptors, GPCRs, and enzymes (ligand binding assay))) EUB0000289c PRCP
Assay data:1 Tested
SummaryRelated BioAssays by Target
Enzyme Activity Assay from US Patent US9365539: "Prolylcarboxypeptidase inhibitors"
Assay data:11 Active, 4 Activity ≤ 1 nM, 11 Activity ≤ 1 µM, 11 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Activation Assay from US Patent US9193762: "Selective inhibitors of prolylcarboxypeptidase"
Assay data:1 Active, 27 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
Enzyme Assay from US Patent US9193762: "Selective inhibitors of prolylcarboxypeptidase"
Assay data:30 Tested
SummaryRelated BioAssays by DepositorRelated BioAssays by Target
Enzyme Activity Assay from US Patent US9006268: "Prolylcarboxypeptidase inhibitors"
Assay data:10 Active, 2 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
Enzyme Activity Assay from US Patent US8785634: "Spiropiperidine prolylcarboxypeptidase inhibitors"
Assay data:9 Active, 2 Activity ≤ 1 nM, 9 Activity ≤ 1 µM, 9 Tested
Enzyme Activity Assay from US Patent US8669252: "Prolylcarboxypeptidase inhibitors"
Assay data:14 Active, 4 Activity ≤ 1 nM, 14 Activity ≤ 1 µM, 14 Tested
Enzyme Activity Assay from US Patent US8569299: "Prolylcarboxypeptidase inhibitors"
Assay data:10 Active, 3 Activity ≤ 1 nM, 10 Activity ≤ 1 µM, 10 Tested
PCP CEREP ligand profiling
PCP Ligand binding assay
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by Target
Inhibition of prolylcarboxypeptidase (unknown origin) at 10 nM to 33.3 uM after 30 mins by gel-based ABPP assay
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Human Prolylcarboxypeptidase (S28: Lysosomal Pro-Xaa carboxypeptidase)
Inhibition of Prcp in mouse Neuro2a cells at 3 nM after 4 hrs by ABPP-SILAC assay
Assay data:3 Tested
SummaryPubMed CitationRelated BioAssays by Target
Inhibition of recombinant mouse PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate after 30 mins by continuous fluorometric assay
Assay data:12 Active, 1 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 12 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate after 30 mins by continuous fluorometric assay
Assay data:25 Active, 24 Activity ≤ 1 µM, 25 Tested
Inhibition of recombinant human PrCP using Mca-Ala-Pro-Lys(Dnp)-OH as substrate measured for 30 mins by fluorescence assay
Assay data:22 Active, 5 Activity ≤ 1 nM, 22 Activity ≤ 1 µM, 22 Tested
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