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Agonist activity at rat GluN1/GluN2D NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode voltage-clamp recording assay
Assay data:11 Active, 7 Activity ≤ 1 µM, 12 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Agonist activity at rat GluN1/GluN2C NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode voltage-clamp recording assay
Assay data:21 Active, 10 Activity ≤ 1 µM, 21 Tested
Agonist activity at rat GluN1/GluN2B NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode voltage-clamp recording assay
Assay data:4 Active, 2 Activity ≤ 1 µM, 4 Tested
Agonist activity at rat GluN1/GluN2A NMDA receptor expressed in Xenopus oocytes measured after 4 days in presence of L-glutamte by two-electrode voltage-clamp recording assay
Assay data:14 Active, 8 Activity ≤ 1 µM, 15 Tested
Membrane potential based assay for SLC6A5 using HEK-293 SLC6A5 OE cells
Assay data:1 Active, 1 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Target
Membrane potential based assay for SLC6A9 using HEK-293 SLC6A9 OE cells
Assay data:1 Active, 2 Tested
Agonist activity at PSGR/OR51E2 (unknown origin) expressed in human Hana3A cells co-transfected with CRE-Luc by luciferase reporter gene assay
Assay data:20 Active, 8 Activity ≤ 1 nM, 20 Activity ≤ 1 µM, 24 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Human GluN2A (Ionotropic glutamate receptors)
Assay data:35 Active, 35 Tested
SummaryCompounds, ActivePubMed CitationRelated BioAssays by Target
Human GluN1 (Ionotropic glutamate receptors)
Assay data:17 Active, 17 Tested
Human GluN2C (Ionotropic glutamate receptors)
Human GluN2B (Ionotropic glutamate receptors)
Assay data:34 Active, 34 Tested
Inhibition of human CYP3A4 assessed as ratio of IC50 in absence of NADPH to IC50 for presence of NADPH using 7-benzyloxyquinoline as substrate after 30 mins
Assay data:155 Active, 221 Tested
Inhibition of human CYP3A4 assessed as ratio of IC50 in absence of NADPH to IC50 for presence of NADPH using diethoxyfluorescein as substrate after 30 mins
Assay data:138 Active, 221 Tested
Inhibition of human CYP2D6 assessed as ratio of IC50 in absence of NADPH to IC50 for presence of NADPH using 4-methylaminoethyl-7-methoxycoumarin as substrate after 30 mins
Assay data:160 Active, 221 Tested
Inhibition of human CYP2C19 assessed as ratio of IC50 in absence of NADPH to IC50 for presence of NADPH using 3-butyryl-7-methoxycoumarin as substrate after 30 mins
Assay data:141 Active, 221 Tested
Inhibition of human CYP2C9 assessed as ratio of IC50 in absence of NADPH to IC50 for presence of NADPH using 7-methoxy-4-trifluoromethylcoumarin-3-acetic acid as substrate after 30 mins
Assay data:163 Active, 221 Tested
Inhibition of human CYP1A2 assessed as ratio of IC50 in absence of NADPH to IC50 for presence of NADPH using ethoxyresorufin as substrate after 30 mins
Assay data:162 Active, 221 Tested
Inhibition of rat glutamate receptor
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed Citation
Displacement of [3H]glycine from strychnine-insensitive glycine recognition site of NMDA receptor in rat brain cortex membrane
Assay data:44 Active, 24 Activity ≤ 1 µM, 65 Tested
Binding affinity to 30 mM pyridoxal-5'-phosphate assessed as formation of PLP-aldimine by ESI-MS analysis
Assay data:5 Active, 5 Tested
SummaryCompounds, ActivePubMed Citation
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