BioAssays, activity concentration at/below 1 uM for PubChem Compound ( - PubChem BioAssay - NCBI

Warning: The NCBI web site requires JavaScript to function. more...

Links from PubChem Compound

Items: 12

Select item 14251951.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Dual specificity testis-specific protein kinase 2

Assay data:2 Active, 2 Activity ≤ 1 µM, 141 Tested

AID:: 1425195

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14251552.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Receptor-interacting serine/threonine-protein kinase 2

Assay data:47 Active, 1 Activity ≤ 1 nM, 35 Activity ≤ 1 µM, 243 Tested

AID:: 1425155

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14251193.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase N3

Assay data:4 Active, 3 Activity ≤ 1 µM, 147 Tested

AID:: 1425119

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14250904.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase NLK

Assay data:9 Active, 7 Activity ≤ 1 µM, 237 Tested

AID:: 1425090

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14249735.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Discoidin domain-containing receptor 2

Assay data:44 Active, 26 Activity ≤ 1 µM, 243 Tested

AID:: 1424973

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14249726.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Epithelial discoidin domain-containing receptor 1

Assay data:52 Active, 37 Activity ≤ 1 µM, 243 Tested

AID:: 1424972

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14249637.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Casein kinase I isoform epsilon

Assay data:17 Active, 6 Activity ≤ 1 µM, 243 Tested

AID:: 1424963

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14249628.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Casein kinase I isoform delta

Assay data:16 Active, 6 Activity ≤ 1 µM, 243 Tested

AID:: 1424962

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 14249229.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Bone morphogenetic protein receptor type-1B

Assay data:12 Active, 6 Activity ≤ 1 µM, 240 Tested

AID:: 1424922

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 142490210.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Activin receptor type-2B

Assay data:7 Active, 3 Activity ≤ 1 µM, 238 Tested

AID:: 1424902

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 142490111.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Activin receptor type-1B

Assay data:16 Active, 1 Activity ≤ 1 nM, 12 Activity ≤ 1 µM, 242 Tested

AID:: 1424901

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 142490012.

Kinobeads (epsilon), multiple immobilized ATP-competitive broad spectrum kinase inhibitors, used to assess residual binding of ~300 proteins simultaneously from cell lysate in the presence of a compound. Quantitative readout performed by mass spectrometry.

Source:: ChEMBL

Protein Target:: Activin receptor type-1

Assay data:21 Active, 13 Activity ≤ 1 µM, 243 Tested

AID:: 1424900

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Supplemental Content

Filters: Manage Filters

Refine your results

• What's this?

BioActivity

Active Compounds (12)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (2)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (12)
BioAssays with the active concentration of tested reagents less than 1 micromolar

Experiment Type

Confirmatory (12)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Depositor Category

Other (12)
BioAssays deposited by other experimentalists

Actions on your results

View or Download BioAssay in PubChem

Find related data

Recent activity

Clear Turn Off Turn On

BioAssays, activity concentration at/below 1 uM for PubChem Compo... (12)
BioAssays, activity concentration at/below 1 uM for PubChem Compound (Select 117606729)
Search

PubChem BioAssay
BioProject Links for BioSample (Select 43929723) (0)
BioProject
Chain A, Natrinema pilin, Orf10
Chain A, Natrinema pilin, Orf10
gi|2563387099|pdb|8GI2|A

Protein
PubChem Compound Links for Structure (Select 249963) (4)
PubChem Compound
protein phosphatase 1 regulatory subunit 3C [Homo sapiens]
protein phosphatase 1 regulatory subunit 3C [Homo sapiens]
gi|4885559|ref|NP_005389.1|

Protein

Your browsing activity is empty.

Activity recording is turned off.

Turn recording back on

See more...

You are here: NCBI > Chemicals & Bioassays > PubChem BioAssay