BioAssays, activity concentration at/below 1 uM for PubChem Compound ( - PubChem BioAssay - NCBI

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Select item 19243951.

Inhibition of recombinant recombinant rat GSK3beta using GS-1 peptide as substrate in presence of [gamma-32P]ATP measured after 30 mins incubation by scintillation counting analysis

Source:: ChEMBL

Protein Target:: Glycogen synthase kinase-3 beta

Assay data:7 Active, 7 Activity ≤ 1 µM, 7 Tested

AID:: 1924395

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 19243942.

Inhibition of recombinant Plasmodium falciparum GSK3 using GS-1 peptide as substrate in presence of [gamma-32P]ATP measured after 30 mins incubation by scintillation counting analysis

Source:: ChEMBL

Assay data:6 Active, 4 Activity ≤ 1 µM, 7 Tested

AID:: 1924394

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953783.

Inhibition of FLT3 (unknown origin)

Source:: ChEMBL

Protein Target:: Receptor-type tyrosine-protein kinase FLT3

Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested

AID:: 1895378

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18953464.

Inhibition of porcine brain GSK-3alpha/beta incubated for 30 mins in presence of [33p]-gamma ATP by scintillation counter analysis

Source:: ChEMBL

Assay data:3 Active, 3 Activity ≤ 1 µM, 5 Tested

AID:: 1895346

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953455.

Inhibition of GST-fused CDK5/p25 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cyclin-dependent kinase 5 activator 1; ...
Total:: 2

Assay data:3 Active, 2 Activity ≤ 1 µM, 5 Tested

AID:: 1895345

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 18953216.

Antiproliferative activity against HUVEC cells assessed as cell growth inhibition measured after 3 days by [3H]-thymidine incorporation assay

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895321

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953207.

Antiangiogenic activity in transgenic zebrafish embryo assessed as inhibition of angiogenic vessel growth incubated for 24 hrs by FITC staining based analysis

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895320

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953178.

Antiproliferative activity against human MV4-11 cells assessed as cell growth inhibition measured after 72 hrs by tetrazolium staining based WST-8 assay

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895317

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 18953169.

Inhibition of recombinant FLT3 D835Y mutant (unknown origin) in presence of ATP by HTRF assay

Source:: ChEMBL

Protein Target:: Receptor-type tyrosine-protein kinase FLT3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895316

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189531510.

Inhibition of recombinant FLT3 (unknown origin) in presence of ATP by HTRF assay

Source:: ChEMBL

Protein Target:: Receptor-type tyrosine-protein kinase FLT3

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895315

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189531111.

Inhibition of SGK (unknown origin) in presence of ATP

Source:: ChEMBL

Protein Target:: Serine/threonine-protein kinase Sgk1

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895311

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189531012.

Inhibition of LCK (unknown origin) in presence of ATP

Source:: ChEMBL

Protein Target:: Tyrosine-protein kinase Lck

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895310

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189530913.

Inhibition of AMPK (unknown origin) in presence of ATP

Source:: ChEMBL

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895309

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 189530814.

Inhibition of GSK3beta (unknown origin) in presence of ATP

Source:: ChEMBL

Protein Target:: Glycogen synthase kinase-3 beta

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895308

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189530715.

Inhibition of GST-fused human CDK2/cyclin A expressed in Escherichia coli using histone H1 as substrate in presence of [33p]-gamma ATP and MgATP

Source:: ChEMBL

Protein Targets:: Cyclin-A2; ...
Total:: 2

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895307

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189530416.

Inhibition of GSK3beta (unknown origin) assessed as decrease in tau phosphorylation at Ser214 residue incubated for 30 mins by Western blot assay

Source:: ChEMBL

Protein Target:: Glycogen synthase kinase-3 beta

Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested

AID:: 1895304

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189529217.

Inhibition of CDK5/p35 (unknown origin)

Source:: ChEMBL

Protein Targets:: Cyclin-dependent kinase 5 activator 1; ...
Total:: 2

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1895292

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189529018.

Inhibition of CDK2/cyclin E (unknown origin)

Source:: ChEMBL

Assay data:3 Active, 2 Activity ≤ 1 µM, 3 Tested

AID:: 1895290

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

Select item 189528919.

Inhibition of CDK2/cyclin A (unknown origin)

Source:: ChEMBL

Protein Targets:: Cyclin-A2; ...
Total:: 2

Assay data:6 Active, 2 Activity ≤ 1 µM, 6 Tested

AID:: 1895289

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation Related BioAssays by Target

Select item 189528820.

Inhibition of starfish oocyte CDK1/Cyclin B using histone H1 as substrate incubated for 10 mins in presence of [gamma-32P]ATP by scintillation counter analysis

Source:: ChEMBL

Assay data:4 Active, 3 Activity ≤ 1 µM, 6 Tested

AID:: 1895288

Summary Compounds, Active Compounds, activity ≤ 1 µM PubMed Citation

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Target

Proteins (8)
BioAssays with protein sequences specified as targets

BioActivity

Active Compounds (69)
BioAssays with compounds reported as biologically active
Activity (IC50, etc) ≤ 1 nM (16)
BioAssays with the active concentration of tested reagents less than 1 nanomolar
Activity (IC50, etc) ≤ 1 µM (69)
BioAssays with the active concentration of tested reagents less than 1 micromolar

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Summary (1)
BioAssays summarizing information from multiple assays for validated chemical probes or small molecule leads
Confirmatory (67)
Low-throughput BioAssays where the activity outcome is based on a dose-response relationship with multiple tested concentrations

Assay Project (13)
BioAssays organized into assay projects based on linkage to Summary assays. Click an project below to retrieve the bioassay list for the project. Click 'All Assay Projects' to retrieve all assay projects represented by Summary assays.

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Literature Extraction (51)
BioAssays extracted from the literature
NIH MLP (17)
BioAssays deposited by the NIH Molecular Libraries Program
Other (1)
BioAssays deposited by other experimentalists

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BioAssays, activity concentration at/below 1 uM for PubChem Compo... (69)
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PubChem BioAssay
txid183514[Organism] (7)
Protein
Mus musculus UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 5 (B...
Mus musculus UDP-Gal:betaGlcNAc beta 1,3-galactosyltransferase, polypeptide 5 (B3galt5), transcript variant 2, mRNA
gi|172073166|ref|NM_001122993.1|

Nucleotide
Proechimys longicaudatus voucher MSB:Mamm:57192 hemoglobine alpha globin subunit...
Proechimys longicaudatus voucher MSB:Mamm:57192 hemoglobine alpha globin subunit (HBA) gene, complete cds
gi|1226042089|gb|MF169895.1|

Nucleotide

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