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Radioligand Displacement Assay from Article 10.1016/j.bbrc.2008.06.050: "ERRgamma tethers strongly bisphenol A and 4-alpha-cumylphenol in an induced-fit manner."
Assay data:3 Active, 3 Activity ≤ 1 µM, 4 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by Target
Competitive Binding Assay from US Patent US9688816: "Polyetherimide compositions and methods for the manufacture and use thereof"
Assay data:11 Active, 1 Activity ≤ 1 nM, 3 Activity ≤ 1 µM, 21 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Target
Agonist activity at ERbeta (unknown origin) expressed in human HeLa cells assessed as transcriptional activation measured after 24 hrs by luciferase reporter gene assay
Assay data:3 Active, 1 Activity ≤ 1 nM, 2 Activity ≤ 1 µM, 7 Tested
Agonist activity at ERalpha (unknown origin) expressed in human HeLa cells assessed as transcriptional activation measured after 24 hrs by luciferase reporter gene assay
Assay data:6 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 7 Tested
Displacement of [3H]17-beta estradiol from GST-fused human recombinant ERbeta ligand binding domain expressed in Escherichia coli BL21alpha cells incubated for 1 hr by liquid scintillation counting method
Assay data:7 Active, 1 Activity ≤ 1 nM, 6 Activity ≤ 1 µM, 7 Tested
Displacement of [3H]17-beta estradiol from GST-fused human recombinant ERalpha ligand binding domain expressed in Escherichia coli BL21alpha cells incubated for 1 hr by liquid scintillation counting method
Binding affinity to GST-tagged human ER alpha ligand-binding domain by TR-FRET assay
Assay data:26 Active, 1 Activity ≤ 1 nM, 24 Activity ≤ 1 µM, 31 Tested
Binding affinity to human ERRgamma
Assay data:2 Active, 2 Activity ≤ 1 µM, 10 Tested
Primary qHTS to identify gynecologic anti-cancer compounds using libraries of approved drugs and bioactive compounds
Assay data:1106 Active, 14 Activity ≤ 1 nM, 6478 Activity ≤ 1 µM, 7578 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by Depositor
Agonist activity at estrogen receptor in human MCF7 cells assessed as ERE-mediated transcriptional activity after 24 hrs by luciferase assay
Assay data:4 Active, 4 Activity ≤ 1 µM, 4 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor beta (ER-beta) signaling pathway
Assay data:113 Active, 4 Activity ≤ 1 nM, 67 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS assay to identify small molecule agonists of the endoplasmic reticulum stress response signaling pathway - cell viability counter screen
Assay data:328 Active, 5 Activity ≤ 1 nM, 337 Activity ≤ 1 µM, 9315 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
qHTS assay to identify small molecule agonists of the NFkB signaling pathway - cell viability counter screen
Assay data:296 Active, 4 Activity ≤ 1 nM, 141 Activity ≤ 1 µM, 9315 Tested
Binding affinity to human ERR gamma
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB
Assay data:3916 Active, 206 Activity ≤ 1 nM, 1830 Activity ≤ 1 µM, 3916 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Target
qHTS assay to identify small molecule antagonists of the peroxisome proliferator-activated receptor delta (PPARd) signaling pathway - cell viability counter screen
Assay data:537 Active, 415 Activity ≤ 1 µM, 9305 Tested
qHTS assay for small molecule activators of the heat shock response signaling pathway - cell viability counter screen
Assay data:410 Active, 2 Activity ≤ 1 nM, 209 Activity ≤ 1 µM, 9305 Tested
qHTS assay for small molecule agonists of the antioxidant response element (ARE) signaling pathway - cell viability counter screen
Assay data:592 Active, 112 Activity ≤ 1 µM, 9305 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway using the BG1 cell line
Assay data:1084 Active, 8 Activity ≤ 1 nM, 330 Activity ≤ 1 µM, 10486 Tested
qHTS assay to identify small molecule agonists of the estrogen receptor alpha (ER-alpha) signaling pathway
Assay data:589 Active, 14 Activity ≤ 1 nM, 591 Activity ≤ 1 µM, 10486 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
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