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Nuclear factor erythroid 2-related factor 2/antioxidant responsive element (Nrf2/ARE) small molecule agonists: luciferase reporter gene qHTS assay in human keratinocytes
Assay data:1099 Active, 1 Activity ≤ 1 nM, 143 Activity ≤ 1 µM, 9667 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMRelated BioAssays by DepositorRelated BioAssays by Same Project
Viability Counterscreen for Primary qHTS for Inhibitors of ATXN expression
Assay data:1940 Active, 33 Activity ≤ 1 nM, 9672 Activity ≤ 1 µM, 397420 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS for Inhibitors of ATXN expression: Summary
SummaryPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
qHTS for Inhibitors of ATXN expression: Validation
Assay data:73 Active, 17 Activity ≤ 1 µM, 1280 Tested
qHTS for Inhibitors of ATXN expression: Validation of Cytotoxic Assay
Assay data:44 Active, 10 Activity ≤ 1 µM, 1280 Tested
SummaryCompounds, ActiveCompounds, activity ≤ 1 µMPubMed CitationRelated BioAssays by DepositorRelated BioAssays by Same Project
USP30 deubiquitinase inhibition: Primary qHTS
Assay data:2500 Active, 47480 Tested
SummaryCompounds, ActiveRelated BioAssays by DepositorRelated BioAssays by Same ProjectRelated BioAssays by Target
UCHL1 deubiquitinase inhibition: Primary qHTS
Assay data:97 Active, 47480 Tested
OTUD3 deubiquitinase inhibition: Primary qHTS
Assay data:334 Active, 47480 Tested
USP28 deubiquitinase inhibition: Primary qHTS
Assay data:1413 Active, 47480 Tested
USP10 deubiquitinase inhibition: Primary qHTS
Assay data:509 Active, 47480 Tested
USP17 deubiquitinase inhibition: Primary qHTS
Assay data:3075 Active, 47480 Tested
USP7 deubiquitinase inhibition: Primary qHTS
Assay data:142 Active, 47480 Tested
USP8 deubiquitinase inhibition: Primary qHTS
Assay data:2010 Active, 47480 Tested
OTUD3 deubiquitinase inhibition: Dose-response Confirmation
Assay data:728 Active, 1869 Tested
UCHL1 deubiquitinase inhibition: Dose-response Confirmation
Assay data:52 Active, 375 Tested
USP28 deubiquitinase inhibition: Dose-response Confirmation
Assay data:1416 Active, 1869 Tested
USP30 deubiquitinase inhibition: Dose-response Confirmation
Assay data:1053 Active, 1869 Tested
USP17 deubiquitinase inhibition: Dose-response Confirmation
Assay data:1187 Active, 1869 Tested
USP10 deubiquitinase inhibition: Dose-response Confirmation
Assay data:529 Active, 1075 Tested
USP8 deubiquitinase inhibition: Dose-response Confirmation
Assay data:233 Active, 1075 Tested
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